SCHEMBL1961907

SCHEMBL1961907

Nc1[nH]c(=S)n(CC2CCCCC2)c(=O)c1N=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CYP3A4 P08684 1/20 0.35
PDE5A O76074 3/20 0.34
PDE4A P27815 2/20 0.34
PDE4B Q07343 2/20 0.34
PDE4C Q08493 2/20 0.34
PDE4D Q08499 2/20 0.34
MTOR P42345 2/20 0.33
CCNB2 O95067 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CCNA1 P78396 1/20 0.33
ATR Q13535 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2484816 0.84 ALDH1A1 (0.35) MEN1KMT2AALDH1A1SMN1; SMN2CYP3A4
SCHEMBL1546118 0.79 ALDH1A1 (0.49) MEN1KMT2AALDH1A1SMN1; SMN2CYP3A4
SCHEMBL7783099 0.78 CASP6 (0.40) MEN1KMT2AALDH1A1SMN1; SMN2CYP3A4
SCHEMBL1958096 0.76 ALDH1A1 (0.40) MEN1KMT2AALDH1A1SMN1; SMN2CYP3A4
SCHEMBL1958336 0.74 KMT2A (0.38) MEN1KMT2AALDH1A1SMN1; SMN2CYP3A4
SCHEMBL7783054 0.74 PDE5A (0.42) MEN1KMT2AALDH1A1PDE5APDE4A
SCHEMBL5860525 0.74 PDE5A (0.42) MEN1KMT2AALDH1A1PDE5APDE4A
SCHEMBL7781023 0.73 PDE5A (0.43) MEN1KMT2AALDH1A1SMN1; SMN2CYP3A4
SCHEMBL1960103 0.71 KMT2A (0.63) MEN1KMT2AALDH1A1SMN1; SMN2CYP3A4
SCHEMBL7776481 0.70 PDE5A (0.43) MEN1KMT2AALDH1A1SMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2332541-A1 Use of thioxanthine derivatives as MPO inhibitors AstraZeneca AB (SE) 2011-06-15 EP disclosed