SCHEMBL7783099

SCHEMBL7783099

Nc1c(N=O)c(=O)n(CC2CCCCC2)c(=S)n1CC1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP6 P55212 1/20 0.40
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
CCNB2 O95067 1/20 0.35
CDK1 P06493 1/20 0.35
CCNB1 P14635 1/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
MTOR P42345 1/20 0.35
CCNA1 P78396 1/20 0.35
ATR Q13535 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35
PDE5A O76074 2/20 0.33
PDE1A P54750 4/20 0.32
PDE1B Q01064 4/20 0.32
PDE1C Q14123 4/20 0.32
NPC1 O15118 1/20 0.32
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5860525 0.85 PDE5A (0.42) MEN1KMT2ACCNB2CDK1CCNB1
SCHEMBL7783054 0.85 PDE5A (0.42) MEN1KMT2ACCNB2CDK1CCNB1
SCHEMBL7781023 0.84 PDE5A (0.43) CASP6MEN1KMT2ACCNB2CDK1
SCHEMBL7783094 0.82 PDE5A (0.35) MEN1KMT2APDE5APDE1APDE1B
SCHEMBL7776481 0.81 PDE5A (0.43) CASP6MEN1KMT2ACCNB2CDK1
SCHEMBL7781030 0.79 PDE5A (0.48) PDE5APDE1APDE1BPDE1CPDE4A
SCHEMBL7783337 0.79 CTSK (0.46) MEN1KMT2APDE5APDE1APDE1B
SCHEMBL2484816 0.78 ALDH1A1 (0.35) MEN1KMT2ACCNB2CDK1CCNB1
SCHEMBL1961907 0.78 MEN1 (0.35) MEN1KMT2ACCNB2CDK1CCNB1
SCHEMBL7776470 0.77 PDE5A (0.48) CASP6MEN1KMT2APDE5AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0775141-B1 PHENYL XANTHINE DERIVATIVES WELLCOME FOUND (GB) 2001-09-26 EP disclosed
US-5776940-A COMPOUNDS FOR TREATMENT OF SEPTIC SHOCK, ANTIINFLAMMATORY AND ANTIALLERGENS GLAXO WELLCOME INC. (US) 1998-07-07 US disclosed