SCHEMBL19620886

SCHEMBL19620886

COc1ccc(C(O)OC)c2ccn(C(C)C)c12

nearest known ligand 0.32

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.31
CYP2D6 P10635 1/20 0.31
ADRA2A P08913 1/20 0.31
ADRA1A P35348 1/20 0.31
MGAM O43451 1/20 0.31
GAA P10253 1/20 0.31
SI P14410 1/20 0.31
MGAM2 Q2M2H8 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
CA7 P43166 1/20 0.31
CA9 Q16790 1/20 0.31
MEN1 O00255 1/20 0.31
MAPK1 P28482 1/20 0.31
BLM P54132 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL929611 0.75 IDO1 (0.44) HTR2CGAAMEN1MAPK1KMT2A
SCHEMBL2594989 0.73 MAPT (0.43) GAACA1CA2CA7CA9
SCHEMBL14345499 0.73 HTR2C (0.33) HTR2CCYP2D6
SCHEMBL2594926 0.72 MAPT (0.38) GAACA1CA2CA7CA9
SCHEMBL8931460 0.69 APLNR (0.33) HTR2CADRA2A
SCHEMBL19564699 0.68 HTR2A (0.41) HTR2CGAACA1CA2CA7
SCHEMBL6203758 0.66 CA1 (0.52) CYP2D6CA1CA2CA7CA9
SCHEMBL22909980 0.58 CES2 (0.47) CYP2D6GAACA9
SCHEMBL2588953 0.57 ADRA2A (0.45) HTR2CCYP2D6ADRA2AADRA1AMEN1
SCHEMBL12075669 0.57 IDO1 (0.50) CA1CA2CA7CA9KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246027-A1 INDOLE DERIVATIVES FOR THE TREATMENT OF CANCER GlaxoSmithKline LLC (US) 2017-11-22 EP disclosed