SCHEMBL19622306

SCHEMBL19622306

CCOC(=O)c1cc(F)c(Oc2ccc(BO)c(CO)c2)c(F)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 1/20 0.37
CA12 O43570 3/20 0.37
CA1 P00915 3/20 0.37
CA2 P00918 3/20 0.37
CA7 P43166 3/20 0.37
CA9 Q16790 3/20 0.37
CA14 Q9ULX7 3/20 0.37
ESR1 P03372 1/20 0.37
ESR2 Q92731 1/20 0.37
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
LMNA P02545 3/20 0.36
CYP1A2 P05177 2/20 0.36
CYP3A4 P08684 1/20 0.36
MAOA P21397 1/20 0.36
MAPT P10636 4/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
CASP3 P42574 1/20 0.36
TRPV1 Q8NER1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19622275 0.78 SCN9A (0.40) CYP1A2
SCHEMBL19622328 0.69 PDE4B (0.44) STSESR1L3MBTL1LMNACYP1A2
SCHEMBL14748413 0.69 PDE4B (0.40) STSCA12CA1CA2CA7
SCHEMBL2528983 0.68 PDE4B (0.66)
SCHEMBL19622200 0.68 MAPT (0.40) CA1CA2L3MBTL1LMNAMAPT
SCHEMBL19622230 0.67 HDAC3 (0.36) MAPTKMT2AHPGDSMN1; SMN2TSHR
SCHEMBL17787354 0.67 KDM4E (0.44) ALDH1A1KDM4E
SCHEMBL1999331 0.66 CA12 (0.60) CA12CA1CA2CA7CA9
SCHEMBL15933217 0.66 LTA4H (0.50) CA1CA2MAOASMN1; SMN2TSHR
SCHEMBL27375655 0.65 CA12 (0.50) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed