SCHEMBL19622337

SCHEMBL19622337

COC(=O)c1ccc(Oc2ccc(C)c(CO)c2)nc1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.50
PDE4B Q07343 1/20 0.45
MAPK1 P28482 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPT P10636 2/20 0.44
GAA P10253 2/20 0.44
ALDH1A1 P00352 3/20 0.43
TDP1 Q9NUW8 1/20 0.41
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
P2RX3 P56373 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
GABRA5 P31644 2/20 0.40
CTSA P10619 1/20 0.40
OPRM1 P35372 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19622338 0.87 LMNA (0.49) LMNAPDE4BMAPK1L3MBTL1KDM4E
SCHEMBL4596324 0.80 LMNA (0.52) LMNAPDE4BMAPK1L3MBTL1KDM4E
SCHEMBL12993276 0.79 LMNA (0.48) LMNAMAPK1L3MBTL1KDM4EALDH1A1
SCHEMBL21656526 0.79 LMNA (0.63) LMNAMAPK1L3MBTL1KDM4EGAA
SCHEMBL23474086 0.78 LMNA (0.52) LMNAPDE4BMAPK1L3MBTL1KDM4E
SCHEMBL12788053 0.77 ALDH1A1 (0.56) LMNAKDM4EMAPTGAAALDH1A1
SCHEMBL21656974 0.77 LMNA (0.60) LMNAMAPK1L3MBTL1KDM4EMAPT
SCHEMBL17176930 0.76 PDE4B (0.53) LMNAPDE4BL3MBTL1KDM4EMAPT
SCHEMBL19808813 0.76 LMNA (0.47) LMNAMAPK1L3MBTL1KDM4EMAPT
SCHEMBL30879440 0.76 LMNA (0.62) LMNAKDM4EMAPTALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed