SCHEMBL19623601

SCHEMBL19623601

CCN(CC)CCNC(=O)c1cccc(-c2nc(N3CCOCC3)nc3c2CCCC3)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 4/20 0.49
HTT P42858 2/20 0.45
TP53 P04637 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
MTOR P42345 2/20 0.43
PIK3CG P48736 2/20 0.43
CAMK2D Q13557 3/20 0.42
USP7 Q93009 2/20 0.41
MAPT P10636 1/20 0.41
GLS O94925 1/20 0.40
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
AKT1 P31749 2/20 0.39
AKT2 P31751 2/20 0.39
AKT3 Q9Y243 2/20 0.39
ADORA2A P29274 1/20 0.39
ADORA1 P30542 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19623572 0.87 PIK3CA (0.49) PIK3CAMEN1KMT2AMTORPIK3CG
SCHEMBL19623865 0.85 PIK3CA (0.50) PIK3CAMEN1KMT2AMTORPIK3CG
SCHEMBL19623703 0.85 PIK3CA (0.49) PIK3CAMEN1KMT2AMTORPIK3CG
SCHEMBL3833880 0.82 PIK3CA (0.75) PIK3CA
SCHEMBL19623871 0.82 PIK3CA (0.47) PIK3CAMTORMAPTKDM4EHPGD
SCHEMBL2378551 0.81 PIK3CA (0.63) PIK3CA
SCHEMBL19623874 0.80 MEN1 (0.48) PIK3CAHTTSMN1; SMN2MEN1KMT2A
SCHEMBL24697994 0.80 PIK3CA (0.45) PIK3CASMN1; SMN2MEN1KMT2AMAPT
SCHEMBL24698899 0.79 PRKD1 (0.42) PIK3CATP53SMN1; SMN2MEN1KMT2A
Trifluoroacetic Acid SCHEMBL2378881 0.78 PIK3CA (0.68) PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed