SCHEMBL19623874

SCHEMBL19623874

O=C(NCC1CCCCC1)c1cccc(-c2nc(N3CCOCC3)nc3c2CCC3)c1

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.48
KMT2A Q03164 3/20 0.48
PIK3CA P42336 2/20 0.48
PDGFRB P09619 1/20 0.45
KDR P35968 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
NAPEPLD Q6IQ20 8/20 0.44
ALDH1A1 P00352 2/20 0.44
HTT P42858 1/20 0.43
POLB P06746 1/20 0.42
LMNA P02545 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MTOR P42345 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19623703 0.84 PIK3CA (0.49) MEN1KMT2APIK3CAALDH1A1MTOR
SCHEMBL19623865 0.83 PIK3CA (0.50) MEN1KMT2APIK3CAPDGFRBKDR
SCHEMBL19623572 0.82 PIK3CA (0.49) MEN1KMT2APIK3CAMTOR
SCHEMBL2378244 0.81 PIK3CA (0.64) PIK3CAPDGFRBKDR
SCHEMBL19623601 0.80 PIK3CA (0.49) MEN1KMT2APIK3CAHTTSMN1; SMN2
SCHEMBL24698899 0.78 PRKD1 (0.42) MEN1KMT2APIK3CASMN1; SMN2MTOR
SCHEMBL19623871 0.78 PIK3CA (0.47) PIK3CAKDRHDAC6ALDH1A1MTOR
SCHEMBL24697994 0.78 PIK3CA (0.45) MEN1KMT2APIK3CASMN1; SMN2
SCHEMBL24697633 0.78 PIK3CA (0.41) MEN1KMT2APIK3CAALDH1A1SMN1; SMN2
SCHEMBL19623886 0.77 PIK3CA (0.49) MEN1KMT2APIK3CAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed