SCHEMBL19624741

SCHEMBL19624741

Cc1cc(C#N)c2cc(C(N)=O)[nH]c2c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
KDM4E B2RXH2 3/20 0.37
RHEB Q15382 1/20 0.36
GRM2 Q14416 1/20 0.36
MAP2K1 Q02750 1/20 0.34
MAOA P21397 1/20 0.34
MAOB P27338 1/20 0.34
POLB P06746 2/20 0.34
BCAT1 P54687 1/20 0.34
HTR1A P08908 4/20 0.33
DRD2 P14416 2/20 0.33
CCNC P24863 1/20 0.33
CDK8 P49336 1/20 0.33
GAA P10253 1/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23148027 0.86 GRIN1 (0.44) NPC1RAB9AKDM4ERHEBGAA
SCHEMBL23147759 0.80 KDM4E (0.50) NPC1RAB9AKDM4EPOLBGAA
SCHEMBL29813016 0.80 KDM4E (0.50) NPC1RAB9AKDM4EPOLBGAA
SCHEMBL18183354 0.79 NPC1 (0.56) NPC1RAB9AKDM4ERHEBMAP2K1
SCHEMBL11457867 0.78 NPC1 (0.41) NPC1RAB9AKDM4ERHEBMAP2K1
SCHEMBL29063172 0.77 SLC9A1 (0.41) KDM4ERHEBMAP2K1BCAT1HTR1A
SCHEMBL24037986 0.75 MAOA (0.40) NPC1RAB9AKDM4EMAOAMAOB
SCHEMBL15506636 0.72 GRIN1 (0.45) KDM4ERHEBGAA
SCHEMBL23148152 0.72 SMYD3 (0.39) NPC1RAB9AKDM4EPOLBDRD2
SCHEMBL29813126 0.72 SMYD3 (0.39) NPC1RAB9AKDM4EPOLBDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2892880-B1 INDOLE CARBOXAMIDE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2017-11-22 EP disclosed