SCHEMBL19631736

SCHEMBL19631736

OC(c1ccccn1)C1(N2CCN(Cc3ccc(OC(F)(F)F)cc3)CC2)CCOCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRCP P42785 6/20 0.47
NR1I2 O75469 1/20 0.47
ALDH1A1 P00352 1/20 0.43
TSHR P16473 1/20 0.43
KCNH2 Q12809 2/20 0.42
DRD4 P21917 2/20 0.41
LMNA P02545 1/20 0.40
MMP1 P03956 1/20 0.40
MMP2 P08253 1/20 0.40
MMP3 P08254 1/20 0.40
MMP9 P14780 1/20 0.40
MMP8 P22894 1/20 0.40
MMP14 P50281 1/20 0.40
CHRM4 P08173 1/20 0.40
NAMPT P43490 1/20 0.40
DRD2 P14416 1/20 0.40
TEAD1 P28347 2/20 0.39
BCHE P06276 1/20 0.39
ACHE P22303 1/20 0.39
BACE1 P56817 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22169574 0.82 ALDH1A1 (0.39) ALDH1A1KCNH2DRD4DRD2
SCHEMBL21233704 0.81 TRPV6 (0.43) ALDH1A1KCNH2
SCHEMBL19631727 0.80 PRCP (0.49) PRCPALDH1A1TSHRKCNH2DRD4
SCHEMBL22169566 0.76 DRD4 (0.53) ALDH1A1DRD4LMNADRD2
SCHEMBL624525 0.75 NR1I2 (0.72) PRCPNR1I2MMP1MMP2MMP3
SCHEMBL21233604 0.75 CHRM2 (0.41) ALDH1A1CHRM4DRD2
SCHEMBL19631833 0.74 SIGMAR1 (0.41) ALDH1A1KCNH2
SCHEMBL19631873 0.73 SIGMAR1 (0.40) ALDH1A1KCNH2DRD4LMNAACHE
SCHEMBL22169548 0.71 SIGMAR1 (0.40) ALDH1A1TSHRKCNH2LMNA
SCHEMBL648176 0.70 PRCP (0.49) PRCPALDH1A1TSHRKCNH2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198339-A1 TETRAHYDROPYRAN AND THIOPYRAN DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-11-23 WO disclosed