SCHEMBL19631835

SCHEMBL19631835

CN(Cc1ccccc1)[C@@H]1CCN(C2(C(O)c3ccccn3)CCOC(C)(C)C2)C1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.35
NPSR1 Q6W5P4 3/20 0.34
KDM4E B2RXH2 2/20 0.34
OPRM1 P35372 2/20 0.34
SIGMAR1 Q99720 2/20 0.34
ATM Q13315 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
AGTR2 P50052 2/20 0.33
KMT2A Q03164 1/20 0.33
UBE2M P61081 1/20 0.33
DCUN1D1 Q96GG9 1/20 0.33
MCHR1 Q99705 2/20 0.33
ALDH1A1 P00352 2/20 0.32
CCR5 P51681 2/20 0.32
HTR1D P28221 1/20 0.32
HTR1B P28222 1/20 0.32
ICMT O60725 1/20 0.31
HTT P42858 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19631833 0.78 SIGMAR1 (0.41) KDM4EOPRM1SIGMAR1KMT2AALDH1A1
SCHEMBL19631875 0.78 OPRM1 (0.38) LMNANPSR1OPRM1SIGMAR1AGTR2
SCHEMBL21221683 0.78 OPRM1 (0.38) LMNANPSR1OPRM1SIGMAR1AGTR2
SCHEMBL21221670 0.78 OPRM1 (0.38) LMNANPSR1OPRM1SIGMAR1AGTR2
SCHEMBL19615078 0.78 OPRM1 (0.38) LMNANPSR1OPRM1SIGMAR1AGTR2
SCHEMBL19632009 0.78 OPRM1 (0.38) LMNANPSR1OPRM1SIGMAR1AGTR2
SCHEMBL19615076 0.78 OPRM1 (0.38) LMNANPSR1OPRM1SIGMAR1AGTR2
SCHEMBL22169548 0.76 SIGMAR1 (0.40) LMNAOPRM1SIGMAR1KMT2AALDH1A1
SCHEMBL19615050 0.74 ALDH1A1 (0.46) LMNANPSR1KDM4EOPRM1SIGMAR1
SCHEMBL19615051 0.74 ALDH1A1 (0.46) LMNANPSR1KDM4EOPRM1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198339-A1 TETRAHYDROPYRAN AND THIOPYRAN DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-11-23 WO disclosed