SCHEMBL19631968

SCHEMBL19631968

c1ccc(C2(N3CCN(Cc4cccnc4)CC3)CCCCCOCC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.48
CHRNA4 P43681 1/20 0.48
TRPV6 Q9H1D0 4/20 0.44
GRIN2D O15399 1/20 0.44
GRIN3B O60391 1/20 0.44
CYP2B6 P20813 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A4 P31645 1/20 0.44
PRCP P42785 1/20 0.44
SLC6A3 Q01959 1/20 0.44
GRIN1 Q05586 1/20 0.44
KCNH2 Q12809 1/20 0.44
GRIN2A Q12879 1/20 0.44
GRIN2B Q13224 1/20 0.44
GRIN2C Q14957 1/20 0.44
GRIN3A Q8TCU5 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
OPRM1 P35372 2/20 0.44
OPRD1 P41143 2/20 0.44
OPRK1 P41145 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19631577 0.89 SIGMAR1 (0.52) GRIN2DGRIN3BCYP2B6SLC6A2SLC6A4
SCHEMBL19631923 0.82 CHRNB2 (0.47) CHRNB2CHRNA4TRPV6OPRM1OPRD1
SCHEMBL19631679 0.82 SIGMAR1 (0.53) GRIN2DGRIN3BCYP2B6SLC6A2SLC6A4
SCHEMBL9129525 0.79 SIGMAR1 (0.65) GRIN2DGRIN3BCYP2B6SLC6A2SLC6A4
Phencyclidine SCHEMBL28206533 0.74 GRIN1 (0.80) GRIN2DGRIN3BCYP2B6SLC6A2SLC6A4
SCHEMBL16111935 0.72 SIGMAR1 (0.62) GRIN2DGRIN3BCYP2B6SLC6A2SLC6A4
SCHEMBL4970159 0.72 CHRNB2 (0.72) CHRNB2CHRNA4TRPV6KDM4EALDH1A1
SCHEMBL15800693 0.72 CHRNB2 (0.77) CHRNB2CHRNA4TRPV6SIGMAR1KDM4E
SCHEMBL7388493 0.71 SIGMAR1 (0.73) GRIN2DGRIN3BCYP2B6SLC6A2SLC6A4
SCHEMBL16026435 0.71 CHRNB2 (0.85) CHRNB2CHRNA4TRPV6KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198339-A1 TETRAHYDROPYRAN AND THIOPYRAN DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-11-23 WO disclosed