SCHEMBL19631577

SCHEMBL19631577

c1ccc(CN2CCN(C3(c4ccccc4)CCCCCOCC3)CC2)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 7/20 0.52
KCNH2 Q12809 2/20 0.52
GRIN2D O15399 1/20 0.52
GRIN3B O60391 1/20 0.52
CYP2B6 P20813 1/20 0.52
SLC6A2 P23975 1/20 0.52
SLC6A4 P31645 1/20 0.52
PRCP P42785 1/20 0.52
SLC6A3 Q01959 1/20 0.52
GRIN1 Q05586 1/20 0.52
GRIN2A Q12879 1/20 0.52
GRIN2B Q13224 1/20 0.52
GRIN2C Q14957 1/20 0.52
GRIN3A Q8TCU5 1/20 0.52
OPRM1 P35372 4/20 0.51
OPRD1 P41143 1/20 0.51
NPSR1 Q6W5P4 1/20 0.45
OPRL1 P41146 1/20 0.45
POLB P06746 1/20 0.44
TMEM97 Q5BJF2 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19631679 0.92 SIGMAR1 (0.53) SIGMAR1KCNH2GRIN2DGRIN3BCYP2B6
SCHEMBL9129525 0.89 SIGMAR1 (0.65) SIGMAR1KCNH2GRIN2DGRIN3BCYP2B6
SCHEMBL19631968 0.89 CHRNB2 (0.48) SIGMAR1KCNH2GRIN2DGRIN3BCYP2B6
SCHEMBL16111935 0.82 SIGMAR1 (0.62) SIGMAR1KCNH2GRIN2DGRIN3BCYP2B6
Phencyclidine SCHEMBL28206533 0.81 GRIN1 (0.80) SIGMAR1KCNH2GRIN2DGRIN3BCYP2B6
SCHEMBL19615068 0.79 NPSR1 (0.44) SIGMAR1KCNH2GRIN2DGRIN3BCYP2B6
SCHEMBL21337174 0.79 SIGMAR1 (0.51) SIGMAR1KCNH2OPRM1TMEM97DRD4
SCHEMBL7317077 0.78 SIGMAR1 (0.65) SIGMAR1KCNH2GRIN2DGRIN3BCYP2B6
SCHEMBL21337177 0.78 OPRM1 (0.46) SIGMAR1KCNH2OPRM1OPRL1TMEM97
SCHEMBL7388493 0.78 SIGMAR1 (0.73) SIGMAR1KCNH2GRIN2DGRIN3BCYP2B6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198339-A1 TETRAHYDROPYRAN AND THIOPYRAN DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-11-23 WO disclosed