SCHEMBL19631996

SCHEMBL19631996

C/C(=N\O)c1cc(C#N)ccn1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.49
GRM4 Q14833 1/20 0.36
LRRK2 Q5S007 1/20 0.36
HTT P42858 1/20 0.35
GRM5 P41594 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
LMNA P02545 1/20 0.34
PYGL P06737 1/20 0.34
PYGM P11217 1/20 0.34
NOS3 P29474 2/20 0.33
NOS1 P29475 2/20 0.33
TRPV4 Q9HBA0 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
PKN1 Q16512 1/20 0.32
PKN2 Q16513 1/20 0.32
ANO1 Q5XXA6 1/20 0.32
RORC P51449 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4946681 0.79 PYGL (0.36) GRM4LRRK2GRM5CLK4PYGL
SCHEMBL1853358 0.79 ALDH1A1 (0.46) KDM4EGRM4LRRK2GRM5CLK4
SCHEMBL3511033 0.79 LRRK2 (0.40) GRM4LRRK2GRM5CLK4PYGL
SCHEMBL19278272 0.76 GRM5 (0.37) KDM4EGRM4HTTGRM5CLK4
SCHEMBL8284487 0.74 KDM4E (0.55) KDM4EMAPTKDM4C
SCHEMBL6840488 0.74 KDM4E (0.55) KDM4EHTTLMNANOS3NOS1
SCHEMBL5936390 0.73 KDM4C (0.55) KDM4EGRM4LRRK2GRM5LMNA
Water SCHEMBL347466 0.73 KDM4C (0.55) KDM4EGRM4LRRK2GRM5LMNA
SCHEMBL16139802 0.73 KDM4E (0.53) KDM4EHTTGRM5LMNAMAPT
SCHEMBL13593104 0.73 KDM4E (0.53) KDM4EGRM5MAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198785-A1 OXIME DERIVATIVES USEFUL AS INHIBITORS OF HISTONE DEMETHYLASE KDM4C IEO - ISTITUTO EUROPEO DI ONCOLOGIA S.R.L. (IT) 2017-11-23 WO disclosed