SCHEMBL19633751

SCHEMBL19633751

COc1cc(COc2ccc3c(Nc4cccc(C(F)(F)F)c4)ccnc3c2)cc(OC)c1OC

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAK O14976 15/20 0.66
RIPK2 O43353 7/20 0.59
COQ8A Q8NI60 7/20 0.59
NLK Q9UBE8 7/20 0.59
EPHB6 O15197 2/20 0.57
ABL1 P00519 2/20 0.57
LCK P06239 2/20 0.57
EPHA1 P21709 2/20 0.57
EPHA8 P29322 2/20 0.57
TXK P42681 1/20 0.57
GSK3A P49840 1/20 0.56
GSK3B P49841 1/20 0.56
EGFR P00533 3/20 0.48
BMPR1B O00238 1/20 0.48
SRC P12931 1/20 0.48
ACVR1 Q04771 1/20 0.48
MAP2K5 Q13163 1/20 0.48
ABCG2 Q9UNQ0 1/20 0.48
LMNA P02545 1/20 0.48
HTT P42858 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633778 0.92 GAK (0.69) GAKRIPK2COQ8ANLKEPHB6
SCHEMBL19633629 0.90 GSK3A (0.61) GAKRIPK2COQ8ANLKEPHB6
SCHEMBL19633780 0.88 GAK (0.71) GAKRIPK2COQ8ANLKEPHB6
SCHEMBL19633777 0.82 GAK (0.57) GAKRIPK2COQ8ANLKEPHB6
SCHEMBL21121558 0.80 GAK (0.68) GAKRIPK2COQ8ANLKEPHB6
SCHEMBL30420604 0.80 GAK (0.68) GAKRIPK2COQ8ANLKEPHB6
SCHEMBL19633699 0.79 GAK (0.57) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633682 0.78 GSK3A (0.52) GAKGSK3AGSK3BKDRCLK2
SCHEMBL19633713 0.78 GAK (0.49) GAKRIPK2COQ8ANLKEPHB6
SCHEMBL19633519 0.77 GAK (0.57) GAKRIPK2COQ8ANLKGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed