SCHEMBL19633760

SCHEMBL19633760

COc1cc(COc2ccc3c(Sc4ccc(F)cc4)ccnc3c2)cc(OC)c1OC

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 3/20 0.48
KDR P35968 2/20 0.48
GAK O14976 7/20 0.47
MET P08581 5/20 0.47
TUBB1 Q9H4B7 4/20 0.46
TUBB4A P04350 3/20 0.46
TUBB P07437 3/20 0.46
TUBA3C P0DPH7 3/20 0.46
TUBA1B P68363 3/20 0.46
TUBA4A P68366 3/20 0.46
TUBB4B P68371 3/20 0.46
TUBB3 Q13509 3/20 0.46
TUBB2A Q13885 3/20 0.46
TUBB8 Q3ZCM7 3/20 0.46
TUBA3E Q6PEY2 3/20 0.46
TUBA1A Q71U36 3/20 0.46
TUBA1C Q9BQE3 3/20 0.46
TUBB6 Q9BUF5 3/20 0.46
TUBB2B Q9BVA1 3/20 0.46
RIPK2 O43353 3/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633753 0.85 GAK (0.49) PDGFRAKDRGAKTUBB1TUBB4A
SCHEMBL19633759 0.84 TUBB1 (0.49) PDGFRAKDRGAKTUBB1TUBB4A
SCHEMBL19633762 0.83 TUBB1 (0.43) PDGFRAKDRGAKTUBB1TUBB4A
SCHEMBL19633698 0.79 TUBB1 (0.57) GAKMETTUBB1TUBB4ATUBB
SCHEMBL19633779 0.77 TUBB1 (0.65) GAKTUBB1TUBB4ATUBBTUBA3C
SCHEMBL19633749 0.77 TUBB1 (0.54) GAKTUBB1TUBB4ATUBBTUBA3C
SCHEMBL19633648 0.75 PDGFRA (0.46) PDGFRAKDR
SCHEMBL7480661 0.72 PDGFRA (0.76) PDGFRAKDRMETEGFRLCK
SCHEMBL19633520 0.72 MAOB (0.46) PDGFRAKDR
SCHEMBL19633697 0.72 GAK (0.53) PDGFRAKDRGAKMETTUBB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed