SCHEMBL19634397

SCHEMBL19634397

CC(C)C(=O)NCc1ccc(C(=O)NCCN2CCNCC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HASPIN Q8TF76 4/20 0.55
HDAC2 Q92769 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49
LMNA P02545 1/20 0.47
NAMPT P43490 2/20 0.47
L3MBTL1 Q9Y468 2/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
HSD17B10 Q99714 1/20 0.46
POLB P06746 1/20 0.46
ALDH1A1 P00352 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
SUV39H1 O43463 1/20 0.45
PRMT1 Q99873 1/20 0.45
SMYD3 Q9H7B4 1/20 0.45
GLA P06280 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14853581 0.87 HASPIN (0.53) HASPINHDAC2HDAC8HDAC6NPSR1
SCHEMBL23471160 0.87 HASPIN (0.55) HASPINHDAC2HDAC8HDAC6NPSR1
SCHEMBL19634405 0.86 NAMPT (0.49) HDAC2HDAC8HDAC6NPSR1LMNA
SCHEMBL19634685 0.86 CD274 (0.62) NAMPTKDM4EPOLBALDH1A1
SCHEMBL15947380 0.85 HASPIN (0.56) HASPINHDAC2HDAC8HDAC6NPSR1
SCHEMBL21015347 0.84 HDAC6 (0.55) HASPINHDAC2HDAC8HDAC6NPSR1
SCHEMBL22064075 0.83 ALDH1A1 (0.61) HDAC2HDAC8HDAC6NPSR1L3MBTL1
SCHEMBL20458250 0.83 HASPIN (0.59) HASPINHDAC2HDAC8HDAC6NPSR1
SCHEMBL12015823 0.82 LMNA (0.70) HDAC2HDAC8HDAC6NPSR1LMNA
SCHEMBL19634691 0.80 HASPIN (0.62) HASPINHDAC2HDAC8HDAC6NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed