SCHEMBL19634428

SCHEMBL19634428

CC(C)C(=O)NCc1ccc(C(=O)N(CCOC(=O)CO)CCOC(=O)CO)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.42
ERCC4 Q92889 1/20 0.42
HDAC1 Q13547 7/20 0.38
TPSAB1 Q15661 2/20 0.36
PLG P00747 1/20 0.36
PRSS1 P07477 1/20 0.36
HDAC6 Q9UBN7 5/20 0.36
KMT2A Q03164 2/20 0.36
EPHX2 P34913 1/20 0.36
NR1H4 Q96RI1 1/20 0.36
PTGES O14684 1/20 0.36
RAB9A P51151 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
NPC1 O15118 2/20 0.35
ST14 Q9Y5Y6 1/20 0.35
ALDH1A1 P00352 1/20 0.35
MEN1 O00255 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
DRD2 P14416 1/20 0.34
DRD3 P35462 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19634396 0.94 ERCC1 (0.38) ERCC1ERCC4HDAC1TPSAB1PLG
SCHEMBL19634408 0.88 ERCC1 (0.40) ERCC1ERCC4HDAC1TPSAB1PLG
SCHEMBL23471107 0.86 KMT2A (0.49) HDAC1HDAC6KMT2AEPHX2NR1H4
SCHEMBL21015966 0.86 ERCC1 (0.41) ERCC1ERCC4KMT2ARAB9ASMN1; SMN2
SCHEMBL19634395 0.85 MLYCD (0.46) ERCC1ERCC4HDAC1HDAC6EPHX2
SCHEMBL19634695 0.83 ERCC1 (0.49) ERCC1ERCC4HDAC1HDAC6KMT2A
SCHEMBL21015207 0.83 HDAC6 (0.50) HDAC1HDAC6KMT2AEPHX2NR1H4
SCHEMBL19634735 0.81 ERCC1 (0.37) ERCC1ERCC4KMT2A
SCHEMBL19634399 0.81 ERCC1 (0.44) ERCC1ERCC4HDAC1HDAC6KMT2A
SCHEMBL23471020 0.81 KMT2A (0.43) HDAC1HDAC6KMT2ARAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed