SCHEMBL19634735

SCHEMBL19634735

COCC(=O)OCCN(CCOC(=O)CO)C(=O)c1cccc(CNC(=O)C(C)C)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.37
ERCC4 Q92889 1/20 0.37
BACE1 P56817 5/20 0.36
APP P05067 3/20 0.35
ROCK2 O75116 1/20 0.35
PPARG P37231 1/20 0.35
MMP13 P45452 1/20 0.35
MEP1B Q16820 4/20 0.35
FNTA P49354 2/20 0.35
FNTB P49356 2/20 0.35
KMT2A Q03164 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA3 P07451 1/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
CA5A P35218 1/20 0.34
CA7 P43166 1/20 0.34
CACNA1C Q13936 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21015966 0.94 ERCC1 (0.41) ERCC1ERCC4BACE1APPROCK2
SCHEMBL23471006 0.89 HDAC3 (0.39) ROCK2MMP13CA12CA1CA2
SCHEMBL21015864 0.88 BACE1 (0.38) BACE1APPROCK2PPARGMMP13
SCHEMBL19634396 0.88 ERCC1 (0.38) ERCC1ERCC4CA12CA1CA2
SCHEMBL21015871 0.86 NR1H4 (0.35) ROCK2MMP13SLC7A5
SCHEMBL23470999 0.85 HDAC3 (0.41) ROCK2MMP13FNTAFNTBCA12
SCHEMBL19634408 0.84 ERCC1 (0.40) ERCC1ERCC4KMT2ACA12CA1
SCHEMBL21015862 0.82 NR1H4 (0.38) ROCK2MMP13CA1CA2CA7
SCHEMBL19634741 0.82 SPR (0.44) ERCC1ERCC4BACE1APPROCK2
SCHEMBL19634428 0.81 ERCC1 (0.42) ERCC1ERCC4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed