SCHEMBL19634571

SCHEMBL19634571

CNC(=O)c1ccc(C(=O)OCCO)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 7/20 0.55
TSHR P16473 4/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
HPGD P15428 1/20 0.52
HTT P42858 1/20 0.52
HDAC2 Q92769 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
ESR1 P03372 2/20 0.47
ALDH1A1 P00352 1/20 0.47
CHRM1 P11229 1/20 0.47
SLC6A2 P23975 1/20 0.47
KDR P35968 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
MMP13 P45452 1/20 0.46
MAPT P10636 1/20 0.46
POLB P06746 1/20 0.45
LMNA P02545 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20267404 0.86 ALDH1A1 (0.66) PLK1TSHRSMN1; SMN2HPGDHTT
SCHEMBL19634288 0.86 PLK1 (0.55) PLK1TSHRSMN1; SMN2HPGDHTT
SCHEMBL26378 0.84 TDP1 (0.56) TSHRSMN1; SMN2ESR1ALDH1A1CHRM1
SCHEMBL1962951 0.83 MAPT (0.58) TSHRSMN1; SMN2HPGDESR1ALDH1A1
Acetone SCHEMBL28904622 0.83 TSHR (0.55) TSHRSMN1; SMN2HPGDESR1ALDH1A1
Lithium SCHEMBL30805733 0.82 TDP1 (0.54) TSHRSMN1; SMN2ESR1ALDH1A1CHRM1
SCHEMBL13292517 0.82 TDP1 (0.54) TSHRSMN1; SMN2ESR1ALDH1A1CHRM1
SCHEMBL19235060 0.82 TDP1 (0.54) TSHRSMN1; SMN2ESR1ALDH1A1CHRM1
SCHEMBL26453328 0.82 TDP1 (0.54) TSHRSMN1; SMN2ESR1ALDH1A1CHRM1
Ethylene Glycol SCHEMBL28198373 0.82 TDP1 (0.54) TSHRSMN1; SMN2ESR1ALDH1A1CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed