SCHEMBL19634288

SCHEMBL19634288

CNC(=O)c1ccc(C(=O)OCCOC)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 7/20 0.55
ABCB11 O95342 1/20 0.54
CYP3A4 P08684 1/20 0.54
ADRA2B P18089 1/20 0.54
OPRD1 P41143 1/20 0.54
SCN5A Q14524 1/20 0.54
TSHR P16473 3/20 0.53
HPGD P15428 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
HTT P42858 1/20 0.52
MAPT P10636 3/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC8 Q9BY41 1/20 0.50
HDAC6 Q9UBN7 1/20 0.50
ALDH1A1 P00352 2/20 0.47
ESR1 P03372 1/20 0.47
CHRM1 P11229 1/20 0.47
SLC6A2 P23975 1/20 0.47
KDR P35968 1/20 0.47
TDP1 Q9NUW8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9969969 0.89 TSHR (0.64) ABCB11CYP3A4ADRA2BOPRD1SCN5A
SCHEMBL16640624 0.87 MAPT (0.60) ABCB11CYP3A4ADRA2BOPRD1SCN5A
SCHEMBL19634571 0.86 PLK1 (0.55) PLK1CYP3A4TSHRHPGDSMN1; SMN2
SCHEMBL20267404 0.86 ALDH1A1 (0.66) PLK1CYP3A4TSHRHPGDSMN1; SMN2
Ammonia Solution, Strong SCHEMBL27753060 0.84 TSHR (0.55) ABCB11CYP3A4ADRA2BOPRD1SCN5A
SCHEMBL9928660 0.83 CYP3A4 (0.66) ABCB11CYP3A4ADRA2BOPRD1SCN5A
SCHEMBL14134604 0.82 HPGD (0.57) ABCB11CYP3A4ADRA2BOPRD1SCN5A
SCHEMBL13258383 0.81 TSHR (0.56) ABCB11CYP3A4ADRA2BOPRD1SCN5A
SCHEMBL11941322 0.81 TSHR (0.56) ABCB11CYP3A4ADRA2BOPRD1SCN5A
SCHEMBL19400961 0.81 ALDH1A1 (0.70) ABCB11CYP3A4ADRA2BOPRD1SCN5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed