SCHEMBL19635389

SCHEMBL19635389

CCCC(C)(C)OC(=O)N1CCN(c2ccc(OCc3nn(C)c(/C=C/CCCCO)c3Br)cc2)CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESRRG P62508 2/20 0.38
ESRRB O95718 1/20 0.38
ESR1 P03372 1/20 0.38
ESRRA P11474 1/20 0.38
LMNA P02545 6/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
NPC1 O15118 1/20 0.35
NR2F2 P24468 1/20 0.35
HTT P42858 1/20 0.35
ME2 P23368 1/20 0.33
ME1 P48163 1/20 0.33
ME3 Q16798 1/20 0.33
ABCB1 P08183 1/20 0.33
CNR1 P21554 2/20 0.33
CNR2 P34972 1/20 0.33
MAPT P10636 9/20 0.32
TSHR P16473 2/20 0.32
HPGD P15428 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19615217 0.92 ESRRB (0.45) ESRRGESRRBESR1ESRRALMNA
SCHEMBL19635385 0.92 ESRRB (0.45) ESRRGESRRBESR1ESRRALMNA
SCHEMBL24378052 0.90 MAPT (0.35) ESRRGESRRBESR1ESRRALMNA
SCHEMBL28656087 0.82 LMNA (0.39) ESRRGESRRBESR1ESRRALMNA
SCHEMBL19635255 0.82 LMNA (0.39) ESRRGESRRBESR1ESRRALMNA
SCHEMBL19634868 0.78 SMN1; SMN2 (0.47) ESRRGESRRBESR1ESRRALMNA
SCHEMBL23251241 0.77 SMN1; SMN2 (0.46) ESRRGESRRBESR1ESRRALMNA
SCHEMBL21802200 0.76 MAPT (0.37) LMNASMN1; SMN2ME2ME1ME3
SCHEMBL21802201 0.76 MAPT (0.37) LMNASMN1; SMN2ME2ME1ME3
SCHEMBL19635047 0.73 SMN1; SMN2 (0.47) ESRRGESRRBESR1ESRRALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2017-11-23 WO disclosed