SCHEMBL19635786

SCHEMBL19635786

CS(=O)(=O)c1ccc(OCc2n[nH]c(CO)c2Br)cc1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 3/20 0.39
CYP4A11 Q02928 3/20 0.39
PTGS2 P35354 3/20 0.35
NR1H4 Q96RI1 1/20 0.35
ENPP2 Q13822 1/20 0.35
GHSR Q92847 1/20 0.35
LOXL2 Q9Y4K0 1/20 0.35
CA12 O43570 3/20 0.35
CA1 P00915 3/20 0.35
CA2 P00918 3/20 0.35
CA9 Q16790 3/20 0.35
CA7 P43166 1/20 0.35
HAO1 Q9UJM8 1/20 0.34
PTPRZ1 P23471 1/20 0.33
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19615980 0.74 PTGS2 (0.36) CYP4F2CYP4A11PTGS2NR1H4ENPP2
SCHEMBL1577607 0.69 CA12 (0.40) CYP4F2CYP4A11PTGS2NR1H4GHSR
SCHEMBL1577718 0.67 NR1H4 (0.43) CYP4F2CYP4A11PTGS2NR1H4GHSR
SCHEMBL1577742 0.67 CA12 (0.40) CYP4F2CYP4A11PTGS2CA12CA1
SCHEMBL24378111 0.66 HCAR2 (0.30)
SCHEMBL1577807 0.66 PTGS2 (0.43) CYP4F2CYP4A11PTGS2CA12CA1
SCHEMBL16231881 0.66 CYP4F2 (0.42) CYP4F2CYP4A11PTGS2NR1H4ENPP2
SCHEMBL19635290 0.65 ALDH1A1 (0.41) PTGS2CA12CA9
SCHEMBL4390921 0.65 ALDH1A1 (0.50) PTGS2ENPP2CA12CA1CA2
SCHEMBL7363412 0.64 ALDH1A1 (0.73)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2017-11-23 WO disclosed