SCHEMBL19635865

SCHEMBL19635865

COCc1[nH]nc(C(=O)O)c1Br

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 14/20 0.59
MAPK1 P28482 2/20 0.33
ALDH1A1 P00352 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
KDM5A P29375 1/20 0.33
KDM5B Q9UGL1 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17224976 0.80 HCAR2 (0.70) HCAR2
SCHEMBL16445518 0.79 HCAR2 (0.53) HCAR2PRKAG1PRKAA1PRKAB1
SCHEMBL24378068 0.73 HCAR2 (0.33) HCAR2
SCHEMBL28543309 0.70 HCAR2 (0.45) HCAR2
SCHEMBL28835653 0.69 HCAR2 (0.47) HCAR2MAPK1ALDH1A1
SCHEMBL19634905 0.67 KDM4E (0.47) HCAR2ALDH1A1
SCHEMBL25240918 0.66 HCAR2 (0.44) HCAR2MAPK1ALDH1A1KDM5AKDM5B
SCHEMBL28542157 0.64 KDM4C (0.53) HCAR2MAPK1ALDH1A1
SCHEMBL19615409 0.64 HCAR2 (0.33) HCAR2MAPK1ALDH1A1
SCHEMBL31082342 0.64 LMNA (0.36) HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2017-11-23 WO disclosed