SCHEMBL1963692

SCHEMBL1963692

CCOC(=O)C1(C)CNC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.47
POLB P06746 1/20 0.46
OPRM1 P35372 2/20 0.40
ATM Q13315 1/20 0.40
ALDH1A1 P00352 2/20 0.39
ALOX15 P16050 2/20 0.38
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
LMNA P02545 2/20 0.37
HSD17B10 Q99714 1/20 0.37
MGAM O43451 1/20 0.36
GAA P10253 1/20 0.36
SI P14410 1/20 0.36
MGAM2 Q2M2H8 1/20 0.36
SOAT1 P35610 1/20 0.36
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL25271505 0.98 BRD4 (0.46) BRD4POLBOPRM1ATMALDH1A1
SCHEMBL15760245 0.84 OPRM1 (0.46) BRD4POLBOPRM1ATMALDH1A1
SCHEMBL2289941 0.81
SCHEMBL5215702 0.81 BRD4 (0.41) BRD4POLBOPRM1ATMALDH1A1
SCHEMBL567321 0.81 BRD4 (0.41) BRD4POLBOPRM1ATMALDH1A1
SCHEMBL567320 0.81 BRD4 (0.41) BRD4POLBOPRM1ATMALDH1A1
SCHEMBL28231627 0.80 ALDH1A1 (0.45) POLBATMALDH1A1LMNAHSD17B10
SCHEMBL3211657 0.80 POLB (0.47) BRD4POLBOPRM1ATMALDH1A1
Hydrochloric Acid SCHEMBL30427479 0.80 BRD4 (0.40) BRD4POLBOPRM1ATMALOX15
Hydrochloric Acid SCHEMBL7093253 0.80 BRD4 (0.40) BRD4POLBOPRM1ATMALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 34 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240327342-A1 COMPOUNDS HAVING S1P5 RECEPTOR AGONISTIC ACTIVITY ONO PHARMACEUTICAL CO., LTD. (JP) 2024-10-03 US disclosed
EP-4431157-A2 1-[[(3S)-3-METHYL-6-(4(4,4-TRIFLUOROBUTOXY)-3,4-DIHYDRONAPHTHALEN-2YL]METHYL]AZETIDINE-3-CARBOXYLIC ACID HAVING S1P5 RECEPTOR AGONIST ACTIVITY FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS AND CANCER ONO Pharmaceutical Co., Ltd. (JP) 2024-09-18 EP disclosed
US-12049445-B2 Compounds having S1P5 receptor agonistic activity ONO PHARMACEUTICAL CO., LTD. (JP) 2024-07-30 US disclosed
CN-111757869-B Compounds having S1P5 receptor agonistic activity 小野药品工业株式会社 2024-03-08 CN disclosed
US-20230066771-A1 NUCLEAR RECEPTOR MODULATORS ABBVIE INC (US) 2023-03-02 US disclosed
US-20220055986-A1 COMPOUNDS HAVING S1P5 RECEPTOR AGONISTIC ACTIVITY ONO PHARMACEUTICAL CO., LTD. (JP) 2022-02-24 US disclosed
US-11198672-B2 Compounds having S1P5 receptor agonistic activity ONO PHARMACEUTICAL CO., LTD. (JP) 2021-12-14 US disclosed
US-20210130293-A1 NUCLEAR RECEPTOR MODULATORS ABBVIE INC (US) 2021-05-06 US disclosed
US-20210087141-A1 COMPOUNDS HAVING S1P5 RECEPTOR AGONISTIC ACTIVITY ONO PHARMACEUTICAL CO., LTD. (JP) 2021-03-25 US disclosed
EP-3757091-A1 COMPOUND HAVING S1P5 RECEPTOR AGONIST ACTIVITY ONO Pharmaceutical Co., Ltd. (JP) 2020-12-30 EP disclosed
WO-2011071570-A1 NOVEL OXADIAZOLE COMPOUNDS ABBOTT LABORATORIES (US) 2011-06-16 WO disclosed
US-7834039-B2 Oxadiazole compounds ABBOTT LABORATORIES (US) 2010-11-16 US disclosed
US-7834039-B2 Oxadiazole compounds ABBOTT LABORATORIES (US) 2010-11-16 US disclosed
US-7834039-B2 Oxadiazole compounds ABBOTT LABORATORIES (US) 2010-11-16 US disclosed
EP-2109364-A1 NOVEL OXADIAZOLE COMPOUNDS Abbott Laboratories (US) 2009-10-21 EP disclosed
US-20080280876-A1 Novel oxadiazole compounds ABBVIE INC. 2008-11-13 US disclosed
US-20080280876-A1 Novel oxadiazole compounds ABBVIE INC. 2008-11-13 US disclosed
US-20080280876-A1 Novel oxadiazole compounds ABBVIE INC. 2008-11-13 US disclosed
WO-2008076356-A1 NOVEL OXADIAZOLE COMPOUNDS ABBOTT LABORATORIES (US) 2008-06-26 WO disclosed
WO-2008076356-A1 NOVEL OXADIAZOLE COMPOUNDS ABBOTT LABORATORIES (US) 2008-06-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12049445-B2 Compounds having S1P5 receptor agonistic activity S1PR5, S1PR1, S1PR4 BRD4 788/4885POLB 3180/4885OPRM1 930/4885
US-20240327342-A1 COMPOUNDS HAVING S1P5 RECEPTOR AGONISTIC ACTIVITY S1PR5, S1PR1, S1PR4 BRD4 788/4885POLB 3180/4885OPRM1 930/4885
US-11198672-B2 Compounds having S1P5 receptor agonistic activity S1PR5, S1PR1, S1PR4 BRD4 788/4885POLB 3180/4885OPRM1 930/4885
US-20210087141-A1 COMPOUNDS HAVING S1P5 RECEPTOR AGONISTIC ACTIVITY S1PR5, S1PR1, S1PR4 BRD4 788/4885POLB 3180/4885OPRM1 930/4885
US-20220055986-A1 COMPOUNDS HAVING S1P5 RECEPTOR AGONISTIC ACTIVITY S1PR5, S1PR1, S1PR4 BRD4 788/4885POLB 3180/4885OPRM1 930/4885
US-20080280876-A1 Novel oxadiazole compounds S1PR3, S1PR1, S1PR2 BRD4 997/4885POLB 4331/4885OPRM1 1382/4885
US-20210130293-A1 NUCLEAR RECEPTOR MODULATORS NR1I2, NR1H2, NR5A2 BRD4 758/4885POLB 3941/4885OPRM1 590/4885
US-20230066771-A1 NUCLEAR RECEPTOR MODULATORS NR1I2, NR1H2, NR5A2 BRD4 758/4885POLB 3941/4885OPRM1 590/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.