SCHEMBL1963835

SCHEMBL1963835

O=C(Cc1ccccc1F)NC(=O)c1cccc2c1C(=O)N(C1CCC(=O)NC1=O)C2

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 16/20 0.54
CSNK1A1 P48729 3/20 0.49
IKZF1 Q13422 1/20 0.49
DDB1 Q16531 4/20 0.43
POLB P06746 2/20 0.41
MAPT P10636 1/20 0.40
IKZF2 Q9UKS7 1/20 0.40
GSPT1 P15170 1/20 0.39
CYP2C19 P33261 1/20 0.39
KCNH2 Q12809 1/20 0.39
USP2 O75604 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1962011 0.89 CRBN (0.53) CRBNCSNK1A1IKZF1DDB1GSPT1
SCHEMBL1962557 0.87 CRBN (0.57) CRBNCSNK1A1IKZF1DDB1POLB
SCHEMBL1962950 0.87 CRBN (0.55) CRBNCSNK1A1IKZF1DDB1POLB
SCHEMBL1962830 0.85 CRBN (0.53) CRBNCSNK1A1IKZF1DDB1POLB
SCHEMBL1963522 0.85 CRBN (0.51) CRBNCSNK1A1IKZF1DDB1POLB
SCHEMBL1962340 0.84 CRBN (0.49) CRBNCSNK1A1IKZF1DDB1GSPT1
SCHEMBL1965760 0.83 CRBN (0.55) CRBNCSNK1A1IKZF1DDB1POLB
SCHEMBL1961959 0.83 CRBN (0.55) CRBNCSNK1A1IKZF1DDB1POLB
SCHEMBL1961754 0.83 CRBN (0.51) CRBNCSNK1A1IKZF1DDB1POLB
SCHEMBL1963723 0.83 CRBN (0.52) CRBNCSNK1A1IKZF1DDB1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US claimed
US-20200113896-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY SIGNAL PHARM LLC (US) 2020-04-16 US disclosed
US-20140314752-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY SIGNAL PHARMACEUTICALS, LLC (US) 2014-10-23 US disclosed
EP-1919892-B1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORP (US) 2013-08-14 EP disclosed
US-8481568-B2 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION (US) 2013-07-09 US disclosed
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SEPRACOR INC. 2011-06-16 US disclosed
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same CELGENE CORPORATION 2007-03-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200113896-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY MTOR, ULK1, RICTOR CRBN 869/4885CSNK1A1 728/4885IKZF1 238/4885
US-20140314752-A1 METHODS FOR TREATING CANCER USING TOR KINASE INHIBITOR COMBINATION THERAPY MTOR, ULK1, RICTOR CRBN 869/4885CSNK1A1 728/4885IKZF1 238/4885
US-20110144158-A1 ISOINDOLE-IMIDE COMPOUNDS AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SI, CYP3A5, CYP2D6 CRBN 2589/4885CSNK1A1 137/4885IKZF1 658/4885
US-20070049618-A1 Isoindole-imide compounds and compositions comprising and methods of using the same SI, CYP3A5, CYP2D6 CRBN 2589/4885CSNK1A1 137/4885IKZF1 658/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.