SCHEMBL19645656

SCHEMBL19645656

COc1cc2c(=O)n(C)cnc2cc1OCc1ccccc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.53
HDAC6 Q9UBN7 2/20 0.52
CTSV O60911 2/20 0.50
CTSL P07711 2/20 0.50
ALDH1A1 P00352 1/20 0.50
POLB P06746 1/20 0.50
EGFR P00533 2/20 0.49
KDM1A O60341 1/20 0.49
TLR9 Q9NR96 1/20 0.48
TLR7 Q9NYK1 1/20 0.48
IRAK1 P51617 1/20 0.48
IRAK4 Q9NWZ3 1/20 0.48
PLK1 P53350 1/20 0.47
KIT P10721 1/20 0.47
KDM4E B2RXH2 1/20 0.47
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
HTT P42858 1/20 0.47
KDR P35968 1/20 0.47
PDPK1 O15530 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4725517 0.85 ELANE (0.50) ELANEHDAC6CTSVCTSLALDH1A1
SCHEMBL4728366 0.84 HDAC6 (0.59) HDAC6ALDH1A1KDM4EHPGD
SCHEMBL6879935 0.83 HDAC6 (0.78) ELANEHDAC6ALDH1A1POLBEGFR
SCHEMBL4781644 0.83 IRAK1 (0.52) ELANEHDAC6CTSVCTSLEGFR
SCHEMBL4594235 0.79 HDAC6 (0.68) HDAC6
SCHEMBL19645642 0.79 HDAC6 (0.52) HDAC6ALDH1A1KDM4E
SCHEMBL7121138 0.78 KIT (0.48) ELANECTSVCTSLALDH1A1POLB
SCHEMBL663991 0.78 HDAC6 (0.54) ELANEHDAC6ALDH1A1POLBEGFR
SCHEMBL4300106 0.78 HDAC6 (0.60) HDAC6ALDH1A1POLBEGFRTLR9
SCHEMBL10296328 0.78 KDM1A (0.56) ELANEEGFRKDM1AIRAK1IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9827248-B2 Therapeutic compounds and uses thereof KALA PHARMACEUTICALS, INC. (US) 2017-11-28 US disclosed