SCHEMBL4725517

SCHEMBL4725517

COc1cc2ncn(C(C)C)c(=O)c2cc1OCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ELANE P08246 1/20 0.50
HDAC6 Q9UBN7 2/20 0.48
CTSV O60911 2/20 0.47
CTSL P07711 2/20 0.47
EGFR P00533 2/20 0.47
KDM1A O60341 1/20 0.47
IRAK1 P51617 1/20 0.46
IRAK4 Q9NWZ3 1/20 0.46
PDE4A P27815 1/20 0.46
PDE4B Q07343 1/20 0.46
PDE4C Q08493 1/20 0.46
PDE4D Q08499 1/20 0.46
ATM Q13315 1/20 0.46
PLK1 P53350 1/20 0.45
KIT P10721 1/20 0.45
ALDH1A1 P00352 1/20 0.45
POLB P06746 1/20 0.45
KDR P35968 1/20 0.45
PDPK1 O15530 1/20 0.45
MET P08581 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19645656 0.85 ELANE (0.53) ELANEHDAC6CTSVCTSLEGFR
SCHEMBL6879935 0.80 HDAC6 (0.78) ELANEHDAC6EGFRPLK1ALDH1A1
SCHEMBL4781644 0.80 IRAK1 (0.52) ELANEHDAC6CTSVCTSLEGFR
SCHEMBL4728780 0.77 PDE10A (0.46) HDAC6ALDH1A1POLBHTT
SCHEMBL663991 0.77 HDAC6 (0.54) ELANEHDAC6EGFRPLK1ALDH1A1
SCHEMBL4594235 0.76 HDAC6 (0.68) HDAC6
SCHEMBL7121138 0.76 KIT (0.48) ELANECTSVCTSLEGFRKDM1A
SCHEMBL4779638 0.75 HDAC6 (0.47) HDAC6EGFRATMHTT
SCHEMBL4300106 0.75 HDAC6 (0.60) HDAC6EGFRALDH1A1POLBLMNA
SCHEMBL10296328 0.75 KDM1A (0.56) ELANEEGFRKDM1AIRAK1IRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008020302-A2 HETEROAROMATIC QUINOLINE-BASED COMPOUNDS AS PHOSPHODIESTERASE (PDE) INHIBITORS PFIZER PRODUCTS INC. (US) 2008-02-21 WO disclosed