SCHEMBL19650271

SCHEMBL19650271

Nc1sc(NC(=O)c2ccc(C(=O)O)s2)nc1-c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.51
RAB9A P51151 4/20 0.51
MEN1 O00255 3/20 0.51
NPSR1 Q6W5P4 2/20 0.51
LMNA P02545 2/20 0.51
PKM P14618 1/20 0.51
ADORA3 P0DMS8 4/20 0.49
ALDH1A1 P00352 5/20 0.48
NPC1 O15118 4/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
KDM4E B2RXH2 2/20 0.46
RXFP1 Q9HBX9 2/20 0.46
ADORA1 P30542 6/20 0.46
ADORA2A P29274 5/20 0.46
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44
XIAP P98170 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21168721 0.90 KMT2A (0.50) KMT2ARAB9AMEN1NPSR1LMNA
SCHEMBL19638277 0.84 SMN1; SMN2 (0.52) KMT2ARAB9AMEN1NPSR1LMNA
SCHEMBL19638183 0.84 KMT2A (0.51) KMT2ARAB9AMEN1NPSR1LMNA
SCHEMBL19638110 0.84 RAB9A (0.51) KMT2ARAB9AMEN1NPSR1LMNA
SCHEMBL544501 0.83 ADORA3 (0.68) KMT2ARAB9AMEN1NPSR1LMNA
SCHEMBL19637993 0.81 ADORA2A (0.65) KMT2ARAB9AMEN1NPSR1LMNA
SCHEMBL24072562 0.80 RAB9A (0.53) KMT2ARAB9AMEN1NPSR1LMNA
SCHEMBL544732 0.79 ALDH1A1 (0.62) KMT2ARAB9AMEN1NPSR1LMNA
SCHEMBL544138 0.76 POLB (0.56) KMT2ARAB9ANPSR1LMNAALDH1A1
SCHEMBL19638078 0.75 KMT2A (0.50) KMT2ARAB9AMEN1NPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3248964-B1 THIAZOLE MODULATORS OF A3 ADENOSINE RECEPTORS PALOBIOFARMA SL (ES) 2019-07-17 EP disclosed
EP-3248964-A1 THIAZOLE MODULATORS OF A3 ADENOSINE RECEPTORS PALOBIOFARMA S.L. (ES) 2017-11-29 EP disclosed