SCHEMBL1966422

SCHEMBL1966422

CC(=O)NOc1ccccc1C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 9/20 0.61
HSD17B10 Q99714 6/20 0.61
HPGD P15428 6/20 0.61
ALDH1A1 P00352 7/20 0.59
ESR1 P03372 1/20 0.59
ITGB3 P05106 1/20 0.59
ITGA2B P08514 1/20 0.59
HMGB1 P09429 1/20 0.59
TSHR P16473 1/20 0.59
GGT1 P19440 1/20 0.59
PTGS1 P23219 1/20 0.59
PTGS2 P35354 1/20 0.59
BLM P54132 1/20 0.59
NAPRT Q6XQN6 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
LMNA P02545 1/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
HTT P42858 2/20 0.51
USP2 O75604 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38660686 1.00 KDM4E (0.61) KDM4EHSD17B10HPGDALDH1A1ESR1
SCHEMBL27762366 0.98 KDM4E (0.59) KDM4EHSD17B10HPGDALDH1A1ESR1
SCHEMBL27784009 0.98 KDM4E (0.59) KDM4EHSD17B10HPGDALDH1A1ESR1
SCHEMBL1130035 0.95 KDM4E (0.56) KDM4EHSD17B10HPGDALDH1A1ESR1
SCHEMBL1129170 0.91 KDM4E (0.51) KDM4EHSD17B10HPGDALDH1A1ESR1
SCHEMBL1129695 0.91 KDM4E (0.51) KDM4EHSD17B10HPGDALDH1A1ESR1
SCHEMBL27762367 0.84 SLC6A3 (0.56) KDM4EHSD17B10HPGDALDH1A1TSHR
SCHEMBL1982429 0.83 KDM4E (0.53) KDM4EHSD17B10HPGDALDH1A1ESR1
SCHEMBL11127664 0.83 KDM4E (0.53) KDM4EHSD17B10HPGDALDH1A1ESR1
SCHEMBL3485366 0.83 KDM4E (0.53) KDM4EHSD17B10HPGDALDH1A1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101538217-B Novel synthesis method of 2-ethoxy-4-amino-5-chlorobenzoic acid and intermediate thereof CHENGDU HONGDA PHARMACEUTICAL CO LTD 2015-04-15 CN claimed
US-4159208-A REACTING ALKALI METAL SALT OF AN AROMATIC CARBOXYLIC ACID AND A METAL SALT IN THE PRESENCE OF CLAY AND ALUMINUM COMPOUND FUJI PHOTO FILM CO., LTD. (JP) 1979-06-26 US claimed
US-20250146074-A1 DETERMINING WHETHER AN IBD PATIENT WILL RESPOND TO 5-ASA THERAPY THE BRIGHAM AND WOMEN'S HOSPITAL, INC. 2025-05-08 US disclosed
CN-108546402-A A kind of preparation method of flame retardant type sealing element rubber material 苏州耐思特塑胶有限公司 2018-09-18 CN disclosed
CN-106883377-A It is a kind of to utilize the curing agent and its method for producing the preparation of TMPTA waste water 苏州顶裕节能设备有限公司 2017-06-23 CN disclosed
CN-101538217-B Novel synthesis method of 2-ethoxy-4-amino-5-chlorobenzoic acid and intermediate thereof CHENGDU HONGDA PHARMACEUTICAL CO LTD 2015-04-15 CN disclosed
CN-103396334-A New synthesis method of 2-ethoxy-4-amino-5-chlorobenzoic acid and intermediate thereof CHENGDU HONGDA PHARMACEUTICAL CO LTD 2013-11-20 CN disclosed
EP-2334178-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF BOWEL DISEASES WITH GRANULATED MESALAMINE Dr. Falk Pharma Gmbh (DE) 2011-06-22 EP disclosed
WO-2010040113-A1 COMPOSITIONS AND METHODS FOR THE TREATMENT OF BOWEL DISEASES WITH GRANULATED MESALAMINE SALIX PHARMACEUTICALS, LTD. (US) 2010-04-08 WO disclosed
CN-101538217-A Novel synthesis method of 2-ethoxy-4-amino-5-chlorobenzoic acid and intermediate thereof CHENGDU KANGHONG PHARMACEUTICA 2009-09-23 CN disclosed
WO-2008044099-A1 CHARGE TRANSFER COMPLEXES IN THE TREATMENT OF INFLAMMATORY BOWEL DISEASES GHISALBERTI CARLO (BR) 2008-04-17 WO disclosed
EP-1409705-B1 A PROCESS FOR THE PRODUCTION OF AN INHIBITOR OF HUMAN PLATELET AGGREGATION AND SOYBEAN LIPOXYGENASE COUNCIL SCIENT IND RES (IN) 2006-05-24 EP disclosed
EP-1409705-A1 A PROCESS FOR THE PRODUCTION OF AN INHIBITOR OF HUMAN PLATELET AGGREGATION AND SOYBEAN LIPOXYGENASE Council of Scientific and Industrial Research;an Indian Reg. body incorporated under Reg. of Societies Act (Act XXI of 1860) (IN) 2004-04-21 EP disclosed
WO-2002074970-A1 A PROCESS FOR THE PRODUCTION OF AN INHIBITOR OF HUMAN PLATELET AGGREGATION AND SOYBEAN LIPOXYGENASE COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2002-09-26 WO disclosed
EP-0145776-A1 A PHARMACEUTICAL COMPOSITION CONTAINING AZO-BIS-SALICYLIC ACID OR A SALT THEREOF AND A METHOD FOR TREATMENT OF INFLAMMATORY CONDITIONS IN THE INTESTINE PHARMACIA AB (SE) 1985-06-26 EP disclosed
WO-1985000012-A1 A PHARMACEUTICAL COMPOSITION CONTAINING AZO-BIS-SALICYLIC ACID OR A SALT THEREOF AND A METHOD FOR TREATMENT OF INFLAMMATORY CONDITIONS IN THE INTESTINE PHARMACIA AB (SE) 1985-01-03 WO disclosed
US-4159208-A REACTING ALKALI METAL SALT OF AN AROMATIC CARBOXYLIC ACID AND A METAL SALT IN THE PRESENCE OF CLAY AND ALUMINUM COMPOUND FUJI PHOTO FILM CO., LTD. (JP) 1979-06-26 US disclosed
US-3954533-A NITROCELLULOSE, NITROGLYCERIN AND BALLISTIC MODIFIERS OF LEAD- AND COPPER- SALTS THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE NAVY (US) 1976-05-04 US disclosed
US-3936451-A Process for producing salts of hexamethylenetetramine UNITED STATES PIPE AND FOUNDRY COMPANY (US) 1976-02-03 US disclosed