SCHEMBL19664255

SCHEMBL19664255

Cc1ccc(-c2nc3cc(NC(=O)CF)ccc3o2)cc1

nearest known ligand 0.70

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 9/20 0.70
POLB P06746 2/20 0.70
RXFP1 Q9HBX9 2/20 0.70
ALDH1A1 P00352 10/20 0.69
HSD17B10 Q99714 10/20 0.69
HPGD P15428 9/20 0.69
SMN1; SMN2 Q16637 7/20 0.69
NPC1 O15118 6/20 0.69
RAB9A P51151 5/20 0.69
THRB P10828 3/20 0.69
TSHR P16473 2/20 0.69
GAA P10253 1/20 0.69
NPSR1 Q6W5P4 1/20 0.69
KDM4E B2RXH2 9/20 0.67
CASP3 P42574 2/20 0.67
SENP8 Q96LD8 2/20 0.67
SENP7 Q9BQF6 2/20 0.67
SENP6 Q9GZR1 2/20 0.67
MAPK1 P28482 1/20 0.65
MAPT P10636 5/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2244672 0.89 CASP3 (0.80) TP53POLBRXFP1ALDH1A1HSD17B10
SCHEMBL2240275 0.87 ALDH1A1 (0.69) TP53POLBRXFP1ALDH1A1HSD17B10
SCHEMBL2245659 0.87 ALDH1A1 (0.87) TP53POLBRXFP1ALDH1A1HSD17B10
SCHEMBL2245254 0.86 ALDH1A1 (0.68) TP53POLBRXFP1ALDH1A1HSD17B10
SCHEMBL2247278 0.85 ALDH1A1 (0.80) TP53POLBRXFP1ALDH1A1HSD17B10
SCHEMBL2245522 0.84 ALDH1A1 (0.68) TP53POLBRXFP1ALDH1A1HSD17B10
SCHEMBL2245490 0.83 TP53 (0.69) TP53POLBRXFP1ALDH1A1HSD17B10
SCHEMBL16217101 0.83 PTGS2 (0.78) TP53POLBRXFP1ALDH1A1HSD17B10
SCHEMBL10016431 0.83 TP53 (1.00) TP53POLBRXFP1ALDH1A1HSD17B10
SCHEMBL2244567 0.82 ALDH1A1 (1.00) TP53POLBRXFP1ALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3251694-A1 DRUG COMBINATIONS FOR THE TREATMENT OF DUCHENNE MUSCULAR DYSTROPHY Summit (Oxford) Limited (GB) 2017-12-06 EP disclosed