SCHEMBL19671027

SCHEMBL19671027

COCCN1CCN(Cc2ccc(C(C)(C)C)cc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.51
SIGMAR1 Q99720 4/20 0.48
KCNH2 Q12809 2/20 0.47
LMNA P02545 1/20 0.47
NR1I2 O75469 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
CNR1 P21554 1/20 0.47
HRH1 P35367 1/20 0.47
OPRK1 P41145 1/20 0.47
PDE4D Q08499 1/20 0.47
GHSR Q92847 1/20 0.47
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
HRH3 Q9Y5N1 2/20 0.46
TEAD1 P28347 2/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
RAB9A P51151 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1044315 0.85 KCNH2 (0.58) KDM4ESIGMAR1KCNH2LMNANR1I2
SCHEMBL24155571 0.84 LMNA (0.46) SIGMAR1LMNAMEN1KMT2AHRH3
SCHEMBL16217371 0.82 KDM4E (0.47) KDM4ESIGMAR1LMNAKMT2AALDH1A1
SCHEMBL17468366 0.82 POLB (0.61) SIGMAR1LMNAMEN1KMT2AHRH3
SCHEMBL21637809 0.82 POLB (0.54) KDM4ESIGMAR1LMNAMEN1KMT2A
SCHEMBL17465264 0.82 KCNH2 (0.53) KDM4ESIGMAR1KCNH2LMNANR1I2
SCHEMBL270535 0.82 LMNA (0.62) KDM4ESIGMAR1KCNH2LMNANR1I2
SCHEMBL16437255 0.81 HRH3 (0.56) KDM4ELMNAHRH3ALDH1A1MAPT
SCHEMBL13020890 0.81 MAPK1 (0.55) KDM4EMAPT
SCHEMBL12203698 0.81 ALDH1A1 (0.59) KDM4ESIGMAR1KCNH2LMNANR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9834521-B2 Choline kinase inhibitors ARIAD PHARMACEUTICALS, INC. (US) 2017-12-05 US disclosed