SCHEMBL270535

SCHEMBL270535

CN1CCN(Cc2ccc(C(C)(C)C)cc2)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.62
MC4R P32245 1/20 0.61
CHKA P35790 4/20 0.59
ALDH1A1 P00352 3/20 0.57
KDM4E B2RXH2 2/20 0.56
MAPT P10636 2/20 0.56
CA2 P00918 1/20 0.56
NCF1 P14598 1/20 0.56
PRMT6 Q96LA8 1/20 0.56
HDAC6 Q9UBN7 1/20 0.55
KCNH2 Q12809 2/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
NR1I2 O75469 1/20 0.52
ADORA3 P0DMS8 1/20 0.52
CNR1 P21554 1/20 0.52
HRH1 P35367 1/20 0.52
OPRK1 P41145 1/20 0.52
PDE4D Q08499 1/20 0.52
GHSR Q92847 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7809477 0.93 CHKA (0.71) LMNAMC4RCHKAALDH1A1KDM4E
SCHEMBL1044315 0.92 KCNH2 (0.58) LMNAALDH1A1KDM4EMAPTKCNH2
SCHEMBL17470856 0.88 KCNH2 (0.49) LMNAMC4RCHKAALDH1A1KDM4E
SCHEMBL17465264 0.86 KCNH2 (0.53) LMNACHKAALDH1A1KDM4EMAPT
SCHEMBL17470847 0.85 ALDH1A1 (0.65) LMNAALDH1A1KDM4EMAPTKCNH2
SCHEMBL10212101 0.85 HRH3 (0.65) ALDH1A1KDM4ENCF1KCNH2MEN1
SCHEMBL797985 0.85 ALDH1A1 (0.59) LMNACHKAALDH1A1KDM4ECA2
SCHEMBL17083366 0.85 HRH3 (0.50) LMNAMC4RCHKAMEN1KMT2A
SCHEMBL12111066 0.84 LMNA (0.57) LMNAMC4RCHKAALDH1A1KDM4E
SCHEMBL12203698 0.84 ALDH1A1 (0.59) LMNAALDH1A1KDM4EMAPTKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 200 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11365196-B2 FGFR inhibitor and application thereof BETTA PHARMACEUTICALS CO., LTD. (CN) 2022-06-21 US disclosed
US-11352343-B2 Urea derivatives and uses thereof KALA PHARMACEUTICALS, INC. (US) 2022-06-07 US disclosed
US-11351168-B1 2,4-disubstituted pyrimidines useful as kinase inhibitors CELGENE CAR LLC (BM) 2022-06-07 US disclosed
US-20210380588-A1 Novel Compounds and Uses Thereof OXFORD FINANCE LLC 2021-12-09 US disclosed
US-20210308121-A1 PRMT5 INHIBITORS AND USES THEREOF Epizyme, Inc. (US) 2021-10-07 US disclosed
US-20210130353-A1 FGFR INHIBITOR AND APPLICATION THEREOF BETTA PHARMACEUTICALS CO., LTD. (CN) 2021-05-06 US disclosed
US-10980794-B2 PRMT5 inhibitors and uses thereof Epizyme, Inc. (US) 2021-04-20 US disclosed
US-10954244-B2 Compounds and uses thereof KALA PHARMACEUTICALS, INC. (US) 2021-03-23 US disclosed
US-20200354367-A1 COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2020-11-12 US disclosed
US-10828300-B2 Substituted 2,4-diaminopyrimidines as kinase inhibitors CELGENE CAR LLC (BM) 2020-11-10 US disclosed
US-20070197537-A1 Heterobicyclic thiophene compounds and methods of use ARRAY BIOPHARMA, INC. 2007-08-23 US disclosed
US-20070191405-A1 Bi-aryl meta-pyrimidine inhibitors of kinases TARGEGEN, INC. (US) 2007-08-16 US disclosed
US-20070161641-A1 Novel heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands AVENTIS PHARMACEUTICALS INC. (US) 2007-07-12 US disclosed
US-20070161641-A1 Novel heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands AVENTIS PHARMACEUTICALS INC. (US) 2007-07-12 US disclosed
US-20070149560-A1 Novel fused triazolones and the uses thereof ASTRAZENECA AB (SE) 2007-06-28 US disclosed
US-20070149560-A1 Novel fused triazolones and the uses thereof ASTRAZENECA AB (SE) 2007-06-28 US disclosed
US-7186724-B2 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands AVENTIS PHARMACEUTICALS INC. (US) 2007-03-06 US disclosed
US-7186724-B2 Heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands AVENTIS PHARMACEUTICALS INC. (US) 2007-03-06 US disclosed
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. 2007-01-04 US disclosed
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling METHYLGENE, INC. 2007-01-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (15 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210308121-A1 PRMT5 INHIBITORS AND USES THEREOF PRMT5, PRMT1, PRMT6 LMNA 2468/4885MC4R 3413/4885CHKA 1140/4885
US-20070197537-A1 Heterobicyclic thiophene compounds and methods of use ERBB2, LCK, SRC LMNA 4174/4885MC4R 2225/4885CHKA 934/4885
US-20200354367-A1 COMPOUNDS AND COMPOSITIONS FOR IRE1 INHIBITION XBP1, RNASE1, ERN1 LMNA 522/4885MC4R 4750/4885CHKA 2013/4885
US-20070191405-A1 Bi-aryl meta-pyrimidine inhibitors of kinases JAK2, TYK2, JAK3 LMNA 4817/4885MC4R 1157/4885CHKA 630/4885
US-20070004675-A1 Inhibitors of VEGF receptor and HGF receptor signaling HGF, MET, FLT1 LMNA 4411/4885MC4R 1384/4885CHKA 2724/4885
US-11351168-B1 2,4-disubstituted pyrimidines useful as kinase inhibitors DCK, CDK2, DTYMK LMNA 4283/4885MC4R 3891/4885CHKA 464/4885
US-11352343-B2 Urea derivatives and uses thereof UACA, RB1, FLT1 LMNA 2477/4885MC4R 1266/4885CHKA 1244/4885
US-11365196-B2 FGFR inhibitor and application thereof FGFR1, FGFR4, FGFR2 LMNA 4231/4885MC4R 1486/4885CHKA 2899/4885
US-20210380588-A1 Novel Compounds and Uses Thereof RB1, VEGFA, UACA LMNA 2524/4885MC4R 176/4885CHKA 922/4885
US-20070149560-A1 Novel fused triazolones and the uses thereof TP53, BRCA1, KLK3 LMNA 3065/4885MC4R 3910/4885CHKA 836/4885
US-10828300-B2 Substituted 2,4-diaminopyrimidines as kinase inhibitors ABL1, DCK, ERBB2 LMNA 4489/4885MC4R 2607/4885CHKA 584/4885
US-10954244-B2 Compounds and uses thereof RB1, VEGFA, FLT4 LMNA 2569/4885MC4R 224/4885CHKA 958/4885
US-20210130353-A1 FGFR INHIBITOR AND APPLICATION THEREOF FGFR1, FGFR4, FGFR2 LMNA 4168/4885MC4R 1343/4885CHKA 3002/4885
US-20070161641-A1 Novel heterocyclic substituted carbonyl derivatives and their use as dopamine D3 receptor ligands DRD3, DRD2, HTR3C LMNA 4087/4885MC4R 465/4885CHKA 2989/4885
US-10980794-B2 PRMT5 inhibitors and uses thereof PRMT5, PRMT1, PRMT6 LMNA 2468/4885MC4R 3413/4885CHKA 1140/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.