SCHEMBL19680002

SCHEMBL19680002

CC[C@@H]1NC(=O)[C@H]([C@H](O)[C@H](C)C/C=C/c2ccc(C(=O)O)cc2)N(C)C(=O)[C@H](C(C)C)N(C)C(=O)C(CC(C)C)N(C)C(=O)[C@H](CC(C)C)N(C)C(=O)[C@@H](C)NC(=O)C(C)NC(=O)[C@H](CC(C)C)N(C)C(=O)C(C(C)C)NC(=O)[C@H](CC(C)C)N(C)C(=O)CN(C)C1=O

nearest known ligand 0.80

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 11/20 0.80
PPIA P62937 5/20 0.80
PPP3CA Q08209 5/20 0.80
PPIB P23284 2/20 0.80
FKBP1B P68106 2/20 0.80
MEN1 O00255 1/20 0.80
NPC1 O15118 1/20 0.80
ABCC3 O15438 1/20 0.80
GMNN O75496 1/20 0.80
USP2 O75604 1/20 0.80
SLCO2B1 O94956 1/20 0.80
ABCB11 O95342 1/20 0.80
LMNA P02545 1/20 0.80
POLB P06746 1/20 0.80
CYP3A4 P08684 1/20 0.80
MAPT P10636 1/20 0.80
RARB P10826 1/20 0.80
CYP2C9 P11712 1/20 0.80
CYP3A5 P20815 1/20 0.80
TACR2 P21452 1/20 0.80

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9979536 1.00 ABCB1 (0.80) ABCB1PPIAPPP3CAPPIBFKBP1B
SCHEMBL21582623 1.00 ABCB1 (0.80) ABCB1PPIAPPP3CAPPIBFKBP1B
SCHEMBL9979647 0.94 PPP3CA (0.80) ABCB1PPIAPPP3CAPPIBFKBP1B
SCHEMBL19680000 0.94 PPP3CA (0.80) ABCB1PPIAPPP3CAPPIBFKBP1B
SCHEMBL13654640 0.93 ABCB1 (0.82) ABCB1PPIAPPP3CAPPIBFKBP1B
SCHEMBL13985971 0.93 ABCB1 (0.82) ABCB1PPIAPPP3CAPPIBFKBP1B
Cyclosporine SCHEMBL1653705 0.92 ABCB1 (0.87) ABCB1PPIAPPP3CAPPIBFKBP1B
Cyclosporine SCHEMBL1653706 0.92 ABCB1 (0.87) ABCB1PPIAPPP3CAPPIBFKBP1B
SCHEMBL13985914 0.92 ABCB1 (0.85) ABCB1PPIAPPP3CAPPIBFKBP1B
SCHEMBL13985911 0.91 ABCB1 (0.77) ABCB1PPIAPPP3CAPPIBFKBP1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170349632-A1 QUINOLIUM CONJUGATES OF CYCLOSPORIN UCL BUSINESS PLC (GB) 2017-12-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170349632-A1 QUINOLIUM CONJUGATES OF CYCLOSPORIN SHMT2, CS, SQOR ABCB1 109/4885PPIA 190/4885PPP3CA 345/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.