SCHEMBL19682190

SCHEMBL19682190

C[C@@H]1NC(=O)[C@H](CCCNC(=N)N)NC(=O)[C@H](CCCNC(=N)N)NC(=O)CNC(=O)CCSSCCNC(=O)[C@H](CO)NC(=O)CNC(=O)CNC1=O

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 5/20 0.39
SIRT1 Q96EB6 5/20 0.39
SIRT3 Q9NTG7 5/20 0.39
CACNA1B Q00975 1/20 0.39
PLAU P00749 1/20 0.37
ITGB3 P05106 1/20 0.37
ITGA2B P08514 1/20 0.37
KDM4A O75164 1/20 0.37
ELANE P08246 4/20 0.37
KLKB1 P03952 1/20 0.37
SIRT7 Q9NRC8 3/20 0.37
SIRT6 Q8N6T7 2/20 0.37
OXTR P30559 1/20 0.37
NNMT P40261 2/20 0.36
PIN1 Q13526 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12518412 0.84 ITGB3 (0.44) SIRT2SIRT1SIRT3ITGB3ITGA2B
SCHEMBL19682189 0.77 KLKB1 (0.45) CACNA1BPLAUITGB3ITGA2BKLKB1
SCHEMBL29666716 0.77 PIN1 (0.46) CACNA1BPLAUITGB3KDM4APIN1
SCHEMBL29569256 0.75 ITGB3 (0.44) SIRT2SIRT1SIRT3CACNA1BITGB3
SCHEMBL29569103 0.75 ITGB3 (0.44) SIRT2SIRT1SIRT3CACNA1BITGB3
SCHEMBL23391095 0.74 OXTR (0.43) SIRT2SIRT1SIRT3ITGB3ITGA2B
SCHEMBL19605445 0.73 ITGB3 (0.55) ITGB3ITGA2B
SCHEMBL24975502 0.72 PIN1 (0.49) ITGB3ITGA2BPIN1
SCHEMBL20982086 0.72 ITGB3 (0.51) CACNA1BITGB3ITGA2B
SCHEMBL23999304 0.72 ITGB3 (0.51) CACNA1BITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017210246-A2 PENICILLAMINE CONJUGATES AND PARTICLES AND FORMULATIONS THEREOF TARVEDA THERAPEUTICS, INC. (US) 2017-12-07 WO disclosed