SCHEMBL19682809

SCHEMBL19682809

O=S(=O)(Cl)c1ccc(Cl)c2cccnc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.54
LMNA P02545 2/20 0.54
HSP90AA1 P07900 2/20 0.54
MAPT P10636 2/20 0.54
BRD4 O60885 1/20 0.54
METAP2 P50579 1/20 0.54
METAP1 P53582 1/20 0.54
SLC40A1 Q9NP59 7/20 0.53
ALDH1A1 P00352 4/20 0.51
CYP3A4 P08684 2/20 0.48
ALOX12 P18054 2/20 0.48
TDP1 Q9NUW8 2/20 0.48
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
RXFP1 Q9HBX9 1/20 0.47
CCR1 P32246 1/20 0.46
CCR8 P51685 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
MMP14 P50281 2/20 0.45
COMT P21964 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL17506546 0.98 KDM4E (0.53) KDM4ELMNAHSP90AA1MAPTBRD4
SCHEMBL22116812 0.86 KDM4E (0.51) KDM4ELMNAHSP90AA1MAPTBRD4
SCHEMBL26920886 0.81 KMT2A (0.51) KDM4EHSP90AA1MAPTSLC40A1ALDH1A1
SCHEMBL16049881 0.81 KDM4E (0.53) KDM4ESLC40A1ALDH1A1L3MBTL1COMT
SCHEMBL22116822 0.79 COMT (0.50) KDM4ELMNAMAPTBRD4SLC40A1
SCHEMBL21596864 0.78 KMT2A (0.52) KDM4ELMNASLC40A1ALDH1A1MEN1
SCHEMBL196536 0.77 KDM4E (0.70) KDM4ELMNAHSP90AA1MAPTBRD4
SCHEMBL19682408 0.76 MAPT (0.60) KDM4ELMNAHSP90AA1MAPTBRD4
SCHEMBL22116653 0.75 ALDH1A1 (0.53) KDM4ELMNAHSP90AA1MAPTALDH1A1
SCHEMBL23379789 0.75 MEN1 (0.50) HSP90AA1SLC40A1ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10889555-B2 Sulfonamide compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2021-01-12 US disclosed
US-20200405697-A1 Antitumor Agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-31 US disclosed
US-20200399235-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-24 US disclosed
EP-3718545-A1 ANTITUMOR AGENT Taiho Pharmaceutical Co., Ltd. (JP) 2020-10-07 EP disclosed
US-20200157066-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-05-21 US disclosed
EP-3466934-A1 SULFONAMIDE COMPOUND OR SALT THEREOF Taiho Pharmaceutical Co., Ltd. (JP) 2019-04-10 EP disclosed
WO-2017209155-A1 SULFONAMIDE COMPOUND OR SALT THEREOF 大鵬薬品工業株式会社 2017-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200399235-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 KDM4E 1551/4885LMNA 3354/4885HSP90AA1 2308/4885
US-20200157066-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 KDM4E 1551/4885LMNA 3354/4885HSP90AA1 2308/4885
US-10889555-B2 Sulfonamide compound or salt thereof RNASEH1, SNRPA1, RRM2 KDM4E 1551/4885LMNA 3354/4885HSP90AA1 2308/4885
US-20200405697-A1 Antitumor Agent HNRNPR, RRM2, RRM2B KDM4E 2851/4885LMNA 3925/4885HSP90AA1 1410/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.