SCHEMBL19682813

SCHEMBL19682813

O=C1CCCc2ccc(S(=O)(=O)Cl)cc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 11/20 0.47
MAOB P27338 11/20 0.47
CYP2A6 P11509 1/20 0.47
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA14 Q9ULX7 1/20 0.43
PRKCI P41743 1/20 0.42
MEN1 O00255 1/20 0.42
MAPK1 P28482 1/20 0.42
KMT2A Q03164 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PBRM1 Q86U86 1/20 0.41
HSD17B1 P14061 1/20 0.38
GRM5 P41594 1/20 0.36
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
RRM1 P23921 1/20 0.36
RRM2B Q7LG56 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6205829 0.89 PBRM1 (0.52) CA12CA1CA2CA7CA14
SCHEMBL29649377 0.83 CA1 (0.66) MAOAMAOBCYP2A6CA12CA1
SCHEMBL7135031 0.83 CA1 (0.66) MAOAMAOBCYP2A6CA12CA1
SCHEMBL6369671 0.82 TDP1 (0.44) MAOAMAOBCA12CA1CA2
SCHEMBL7194507 0.80 BCHE (0.39) MAOACA12CA1CA2CA7
SCHEMBL1546679 0.80 CA12 (0.66) CA12CA1CA2CA7CA14
SCHEMBL29437178 0.80 CA12 (0.66) CA12CA1CA2CA7CA14
SCHEMBL315066 0.79 MAOA (0.51) MAOAMAOBCYP2A6NPSR1GRM5
SCHEMBL10118335 0.78 CA12 (0.58) CA12CA1CA2CA7CA14
SCHEMBL315222 0.78 HTR2C (0.52) MAOAMAOBCYP2A6CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10889555-B2 Sulfonamide compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2021-01-12 US disclosed
US-20200405697-A1 Antitumor Agent TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-31 US disclosed
US-20200399235-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-12-24 US disclosed
EP-3718545-A1 ANTITUMOR AGENT Taiho Pharmaceutical Co., Ltd. (JP) 2020-10-07 EP disclosed
US-20200157066-A1 Sulfonamide Compound or Salt Thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2020-05-21 US disclosed
EP-3466934-A1 SULFONAMIDE COMPOUND OR SALT THEREOF Taiho Pharmaceutical Co., Ltd. (JP) 2019-04-10 EP disclosed
WO-2017209155-A1 SULFONAMIDE COMPOUND OR SALT THEREOF 大鵬薬品工業株式会社 2017-12-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200399235-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 MAOA 2194/4885MAOB 2022/4885CYP2A6 2396/4885
US-20200157066-A1 Sulfonamide Compound or Salt Thereof RNASEH1, SNRPA1, RRM2 MAOA 2194/4885MAOB 2022/4885CYP2A6 2396/4885
US-10889555-B2 Sulfonamide compound or salt thereof RNASEH1, SNRPA1, RRM2 MAOA 2194/4885MAOB 2022/4885CYP2A6 2396/4885
US-20200405697-A1 Antitumor Agent HNRNPR, RRM2, RRM2B MAOA 3262/4885MAOB 3077/4885CYP2A6 3134/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.