SCHEMBL19683824

SCHEMBL19683824

COc1cc(Nc2ccc(Nc3ncnc(N)c3C(=N)c3ccc(OCCN4CCOCC4)cc3)cc2)cc(OC)c1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 4/20 0.47
EGFR P00533 8/20 0.44
ERBB2 P04626 3/20 0.44
KDR P35968 5/20 0.44
EPHA2 P29317 1/20 0.44
EPHB4 P54760 1/20 0.44
HDAC1 Q13547 2/20 0.44
ILK Q13418 1/20 0.43
AURKA O14965 1/20 0.42
ROCK2 O75116 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LCK P06239 1/20 0.42
FYN P06241 1/20 0.42
RET P07949 1/20 0.42
MET P08581 1/20 0.42
MAPT P10636 1/20 0.42
PDGFRA P16234 1/20 0.42
LTK P29376 1/20 0.42
TTK P33981 1/20 0.42
MAP2K2 P36507 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23047300 0.88 ERBB2 (0.47) SRCEGFRERBB2ILKALDH1A1
SCHEMBL19683692 0.87 ERBB2 (0.45) SRCEGFRERBB2KDREPHA2
SCHEMBL19683782 0.83 EGFR (0.45) SRCEGFRERBB2ILKAURKA
SCHEMBL19683608 0.80 EGFR (0.40) SRCEGFRERBB2ILKAURKA
SCHEMBL19683604 0.80 EPHX2 (0.49) EGFRERBB2KDRAURKALCK
SCHEMBL20878942 0.80 EGFR (0.45) SRCEGFRERBB2KDRILK
SCHEMBL20878968 0.79 SRC (0.44) SRCEGFRERBB2KDRHDAC1
SCHEMBL19683816 0.79 EGFR (0.42) SRCEGFRERBB2KDRAURKA
SCHEMBL20878979 0.79 ERBB2 (0.40) SRCEGFRERBB2KDRHDAC1
SCHEMBL20878890 0.79 BRD4 (0.45) HDAC1RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017206962-A1 NOVEL INHIBITOR FOR FLT3 KINASE AND USES THEREOF 合肥中科普瑞昇生物医药科技有限公司 2017-12-07 WO disclosed