SCHEMBL1968455

SCHEMBL1968455

CC(C)(C)N[C@@H]1CCN(C(=O)O)C[C@H]1c1cc(Cl)cc(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
STS P08842 2/20 0.36
NOTUM Q6P988 1/20 0.35
SPTLC2 O15270 5/20 0.35
EPHX2 P34913 1/20 0.34
KCNH2 Q12809 5/20 0.34
CACNA1H O95180 3/20 0.34
CYP2D6 P10635 3/20 0.34
CACNA1I Q9P0X4 3/20 0.33
CCR1 P32246 1/20 0.33
SPR P35270 1/20 0.33
KDM1A O60341 1/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
ADAMTS5 Q9UNA0 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20262220 0.83 RORC (0.44) SPTLC2EPHX2KDM1AMAOAMAOB
SCHEMBL4156476 0.76 NOTUM (0.43) NOTUMSPRADAMTS5
SCHEMBL4156475 0.76 NOTUM (0.43) NOTUMSPRADAMTS5
SCHEMBL1972533 0.75 TLR2 (0.43) KDM1AMAOAMAOB
SCHEMBL1969431 0.75 TLR2 (0.43) KDM1AMAOAMAOB
SCHEMBL4157819 0.75 RHOC (0.43) SPTLC2KCNH2CACNA1I
SCHEMBL4157818 0.75 RHOC (0.43) SPTLC2KCNH2CACNA1I
SCHEMBL1969992 0.73 TACR1 (0.44) CYP2D6
SCHEMBL2247004 0.73 FPR1 (0.45) EPHX2KDM1AMAOAMAOB
SCHEMBL1971251 0.72 SLC6A4 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME TAKEDA PHARMACEUTICAL COMPANY LIMITED 2011-07-21 US disclosed
EP-2336105-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME Takeda Pharmaceutical Company Limited (JP) 2011-06-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110178060-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND USE OF SAME NTSR2, BDKRB1, AVPR1B STS 2213/4885NOTUM 2970/4885SPTLC2 4574/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.