SCHEMBL1968590

SCHEMBL1968590

C=Cc1ccc(-c2nnc(NC(=O)c3ccccc3)s2)c(C)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.54
TP53 P04637 2/20 0.54
PTGER3 P43115 1/20 0.53
NPC1 O15118 7/20 0.50
RAB9A P51151 7/20 0.50
KMT2A Q03164 6/20 0.50
ALDH1A1 P00352 5/20 0.50
MEN1 O00255 5/20 0.50
KDM4E B2RXH2 5/20 0.50
RXFP1 Q9HBX9 3/20 0.50
CSNK2A2 P19784 1/20 0.50
CSNK2A1 P68400 1/20 0.50
MAPK1 P28482 1/20 0.50
HSD17B10 Q99714 2/20 0.48
GLA P06280 1/20 0.48
LMNA P02545 1/20 0.47
HPGD P15428 1/20 0.47
PPARG P37231 1/20 0.47
NCOA2 Q15596 1/20 0.47
NCOA1 Q15788 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1964640 0.90 SMN1; SMN2 (0.55) SMN1; SMN2TP53PTGER3NPC1RAB9A
SCHEMBL1968945 0.81 CSNK2A2 (0.71) SMN1; SMN2TP53NPC1RAB9AKMT2A
SCHEMBL15789035 0.75 MAPT (0.62) TP53NPC1RAB9AKMT2AMEN1
SCHEMBL1968589 0.74 ALDH1A1 (0.40) PTGER3NPC1RAB9AALDH1A1KDM4E
SCHEMBL1966407 0.73 CSNK2A2 (0.60) SMN1; SMN2TP53NPC1RAB9AKMT2A
SCHEMBL1965024 0.72 CSNK2A2 (0.73) SMN1; SMN2TP53NPC1RAB9AKMT2A
SCHEMBL11480689 0.72 CSNK2A2 (0.83) SMN1; SMN2TP53NPC1RAB9AKMT2A
SCHEMBL1488483 0.71 GSK3B (0.37) SMN1; SMN2PTGER3NPC1RAB9AKMT2A
SCHEMBL17318711 0.69 NPC1 (0.69) SMN1; SMN2TP53PTGER3NPC1RAB9A
SCHEMBL12039939 0.69 NPC1 (0.48) SMN1; SMN2TP53NPC1RAB9AKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334670-A1 NEW 2-AMIDOTHIADIAZOLE DERIVATIVES Almirall S.A. (ES) 2011-06-22 EP disclosed