SCHEMBL19685928

SCHEMBL19685928

Cc1ccc2c(c1)-c1ccccc1Oc1ccccc1-c1cc(C)ccc1N2c1ccc2c(=O)n(-c3ccccc3)cc(C)c2c1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 1/20 0.35
ESRRA P11474 1/20 0.35
ESR2 Q92731 1/20 0.35
KDM4E B2RXH2 4/20 0.33
TDO2 P48775 1/20 0.33
IDO2 Q6ZQW0 1/20 0.33
AGTR1 P30556 1/20 0.33
ALDH1A1 P00352 5/20 0.33
HPGD P15428 2/20 0.33
CYP1A2 P05177 1/20 0.33
BLM P54132 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GAA P10253 1/20 0.32
LMNA P02545 5/20 0.32
TP53 P04637 3/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
MAPT P10636 1/20 0.32
CDK8 P49336 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19685930 0.92 ESR1 (0.38) ESR1ESRRAESR2KDM4ETDO2
SCHEMBL19685880 0.90 LMNA (0.38) ESR1ESRRAESR2KDM4ETDO2
SCHEMBL19686086 0.88 BRD4 (0.40) TDO2IDO2AGTR1GAALMNA
SCHEMBL19686363 0.85 MIF (0.33) KDM4ETDO2IDO2AGTR1ALDH1A1
SCHEMBL19685933 0.83 ESR1 (0.32) ESR1ESRRAESR2KDM4EALDH1A1
SCHEMBL19685927 0.80 ESR1 (0.35) ESR1ESRRAESR2KDM4ETDO2
SCHEMBL19685990 0.79 KDM4E (0.31) KDM4EALDH1A1HPGDCYP1A2BLM
SCHEMBL19686085 0.78 BRD4 (0.43) MEN1KMT2A
SCHEMBL19685934 0.78 ESR1 (0.34) ESR1ESRRAESR2KDM4EALDH1A1
SCHEMBL19686088 0.78 BRD4 (0.38) KDM4ETDO2IDO2ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170352817-A1 POLYCYCLIC COMPOUND AND ORGANIC ELECTROLUMINESCENCE DEVICE INCLUDING THE SAME KYUSHU UNIVERSITY, NATIONAL UNIVERSITY CORPORATION (JP) 2017-12-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170352817-A1 POLYCYCLIC COMPOUND AND ORGANIC ELECTROLUMINESCENCE DEVICE INCLUDING THE SAME CYC1, CCNA1, CYCS ESR1 503/4885ESRRA 1108/4885ESR2 808/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.