SCHEMBL19688

SCHEMBL19688

CC(C)(C)OC(=O)N1CCN(c2ccc(C(O)(C(F)(F)F)C(F)(F)F)cc2)[C@@H](CO)C1

nearest known ligand 0.53

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
RORC P51449 13/20 0.53
GCKR Q14397 5/20 0.43
GPR119 Q8TDV5 1/20 0.41
MAPT P10636 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18549 0.92 RORC (0.53) RORCGCKRGPR119MAPT
SCHEMBL12090314 0.89 GPR119 (0.40) RORCGPR119MAPT
SCHEMBL18572 0.86 RORC (0.56) RORCGCKRGPR119
SCHEMBL21360346 0.85 GRM5 (0.42) GPR119MAPT
SCHEMBL20078 0.85 RORC (0.54) RORCGCKR
SCHEMBL19271 0.85 RORC (0.47) RORCGCKR
SCHEMBL16870 0.84 GCKR (0.46) RORCGCKR
SCHEMBL6719383 0.84 GPR119 (0.43) GPR119MAPT
SCHEMBL6719421 0.84 GPR119 (0.43) GPR119MAPT
SCHEMBL15202872 0.84 RORC (0.45) RORCGCKR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027261-A1 SULFONYLPIPERAZINE DERIVATIVES THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN FOR THE TREATMENT OF DIABETES AMGEN INC. (US) 2012-03-01 WO disclosed