SCHEMBL1969115

SCHEMBL1969115

CCOC(=O)c1ccc(-n2cccn2)cc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 1/20 0.53
JAK3 P52333 1/20 0.53
ALDH1A1 P00352 6/20 0.50
HSD17B10 Q99714 1/20 0.50
HPGD P15428 3/20 0.46
RAB9A P51151 3/20 0.46
TSHR P16473 3/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
HTT P42858 1/20 0.45
RXFP1 Q9HBX9 1/20 0.44
NPC1 O15118 3/20 0.43
TP53 P04637 1/20 0.43
LMNA P02545 1/20 0.43
KDM4E B2RXH2 1/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 2/20 0.42
MEN1 O00255 1/20 0.42
USP2 O75604 1/20 0.42
POLB P06746 1/20 0.42
NLRP3 Q96P20 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7419149 0.90 JAK2 (0.53) JAK2JAK3ALDH1A1HSD17B10HPGD
SCHEMBL14130143 0.87 JAK2 (0.53) JAK2JAK3ALDH1A1HPGDRAB9A
SCHEMBL5063232 0.84 JAK2 (0.50) JAK2JAK3ALDH1A1RAB9ATSHR
SCHEMBL1316699 0.82 GPR119 (0.43) JAK2JAK3ALDH1A1RXFP1LMNA
SCHEMBL18094323 0.82 JAK2 (0.51) JAK2JAK3ALDH1A1RAB9ATSHR
SCHEMBL9010477 0.81 JAK2 (0.50) JAK2JAK3ALDH1A1HSD17B10HPGD
SCHEMBL27989056 0.81 LRRK2 (0.39) JAK2JAK3ALDH1A1HSD17B10TSHR
SCHEMBL12121348 0.80 LMNA (0.49) ALDH1A1HSD17B10HPGDLMNAKDM4E
SCHEMBL7415910 0.79 JAK2 (0.48) JAK2JAK3ALDH1A1HPGDRAB9A
SCHEMBL1363765 0.79 RXFP1 (0.61) JAK2JAK3ALDH1A1HPGDRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334683-A1 SATURATED BICYCLIC HETEROCYCLIC DERIVATIVES AS SMO ANTAGONISTS Istituto di ricerche di Biologia Molecolare P. Angeletti S.R.L. (IT) 2011-06-22 EP disclosed
WO-2010023480-A1 SATURATED BICYCLIC HETEROCYCLIC DERIVATIVES AS SMO ANTAGONISTS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2010-03-04 WO disclosed