SCHEMBL19701944

SCHEMBL19701944

CC(=O)N1C[C@@H](C)N(c2cccc(C(C)C)c2)[C@@H](C)C1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.52
PIK3CD O00329 5/20 0.44
CHRM1 P11229 1/20 0.40
HPGD P15428 2/20 0.38
AR P10275 1/20 0.38
PIK3CA P42336 1/20 0.37
PIK3CB P42338 1/20 0.37
PIK3CG P48736 1/20 0.37
LPAR5 Q9H1C0 2/20 0.36
LMNA P02545 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MDM4 O15151 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
TP53 P04637 1/20 0.36
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
TYR P14679 1/20 0.36
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19701955 0.83 NOTUM (0.52) NOTUMPIK3CDHPGDLMNAKDM4E
SCHEMBL19710898 0.81 AR (0.52) NOTUMARLMNAALDH1A1TP53
SCHEMBL19702012 0.81 NOTUM (0.55) NOTUMPIK3CDHPGDSMN1; SMN2ADAM10
SCHEMBL19701947 0.81 PIK3CD (0.38) NOTUMPIK3CDCHRM1ARLMNA
SCHEMBL19701948 0.80 PIK3CD (0.40) NOTUMPIK3CDHPGDKDM4E
SCHEMBL19690264 0.80 ALOX5 (0.45) PIK3CDHPGDARPIK3CAPIK3CB
SCHEMBL19690265 0.80 ALOX5 (0.45) PIK3CDHPGDARPIK3CAPIK3CB
SCHEMBL19701945 0.80 PIK3CD (0.39) NOTUMPIK3CDCHRM1
SCHEMBL19703395 0.80 PIK3CD (0.48) NOTUMPIK3CD
SCHEMBL19701956 0.78 NOTUM (0.55) NOTUMPIK3CDHPGDKDM4EMDM4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20170355707-A1 BICYCLIC HETEROARYL AMINE COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2017-12-14 US disclosed
US-20170355707-A1 BICYCLIC HETEROARYL AMINE COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2017-12-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170355707-A1 BICYCLIC HETEROARYL AMINE COMPOUNDS PIK3R3, JAK2, JAK3 NOTUM 3221/4885PIK3CD 14/4885CHRM1 955/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.