SCHEMBL19733035

SCHEMBL19733035

CC(C)(C)[Si](C)(C)OCC1C=CC(=O)CN1C(=O)O

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DUT P33316 3/20 0.36
NLRP3 Q96P20 2/20 0.33
TOP2A P11388 2/20 0.33
FKBP1A P62942 1/20 0.33
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28699542 1.00 DUT (0.36) DUTNLRP3TOP2AFKBP1ANFKB1
SCHEMBL15320368 0.86 ALDH1A1 (0.38) DUTTOP2AFKBP1ANFKB1NFKB2
SCHEMBL15320366 0.86 ALDH1A1 (0.38) DUTTOP2AFKBP1ANFKB1NFKB2
SCHEMBL15957013 0.80 DUT (0.36) DUTTOP2AFKBP1A
SCHEMBL3628010 0.80 DUT (0.36) DUTTOP2AFKBP1A
SCHEMBL3739744 0.80 DUT (0.36) DUTTOP2AFKBP1A
SCHEMBL28710557 0.79 DUT (0.34) DUTTOP2AFKBP1A
SCHEMBL28710556 0.79 DUT (0.34) DUTTOP2AFKBP1A
SCHEMBL19733026 0.78 FKBP1A (0.32) DUTTOP2AFKBP1A
SCHEMBL19733021 0.76 FKBP1A (0.32) DUTTOP2AFKBP1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2834239-B1 HETEROBICYCLIC COMPOUNDS AS BETA-LACTAMASE INHIBITORS ENTASIS THERAPEUTICS LTD (GB) 2017-12-27 EP disclosed