SCHEMBL19737518

SCHEMBL19737518

Cc1sc2nc(-c3ccncc3)ccc2c1N

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 13/20 0.56
TP53 P04637 5/20 0.56
THRB P10828 1/20 0.56
POLB P06746 3/20 0.54
ROCK2 O75116 1/20 0.54
ROCK1 Q13464 1/20 0.54
CLK4 Q9HAZ1 1/20 0.54
TDP1 Q9NUW8 2/20 0.50
NPC1 O15118 6/20 0.46
RAB9A P51151 6/20 0.46
LIMK1 P53667 3/20 0.46
KDM4E B2RXH2 5/20 0.45
SMN1; SMN2 Q16637 4/20 0.45
HPGD P15428 2/20 0.45
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
NFKB1 P19838 2/20 0.44
NFKB2 Q00653 2/20 0.44
RELA Q04206 2/20 0.44
TLR9 Q9NR96 3/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19805090 0.86 NPC1 (0.61) MAPTTP53THRBPOLBROCK2
SCHEMBL18537683 0.82 LIMK1 (0.67) MAPTTP53THRBPOLBNPC1
SCHEMBL23009514 0.78 KDM4E (0.58) MAPTTP53THRBPOLBROCK2
SCHEMBL20731005 0.74 ALDH1A1 (0.62) MAPTTP53NPC1RAB9ALIMK1
SCHEMBL24729646 0.74 ALDH1A1 (0.45) MAPTTP53POLBNPC1RAB9A
SCHEMBL21051652 0.72 MAP2K3 (0.45) MAPTTP53THRBPOLBROCK2
SCHEMBL19737752 0.72 MAPT (0.85) MAPTTP53THRBPOLBROCK2
SCHEMBL23938107 0.71 KDM4E (0.42) MAPTTP53THRBPOLBTDP1
SCHEMBL8143280 0.69 PIK3CD (0.53) MAPTTP53THRBPOLBROCK2
SCHEMBL23937997 0.69 KDM4E (0.41) MAPTTHRBPOLBTDP1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017217439-A1 THIENO[2,3-b]PYRIDINE DERIVATIVE AND QUINOLINE DERIVATIVE, AND USE THEREOF 国立大学法人東京大学 2017-12-21 WO disclosed