SCHEMBL19737553

SCHEMBL19737553

O=Cc1ccc2c(c1)c(Br)cn2S(=O)(=O)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 11/20 0.49
KDM4E B2RXH2 1/20 0.48
UBE2N P61088 1/20 0.48
AKR1C3 P42330 1/20 0.47
AKR1C1 Q04828 1/20 0.47
CA12 O43570 2/20 0.46
CA9 Q16790 2/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PLK1 P53350 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
HDAC3 O15379 1/20 0.43
HDAC4 P56524 1/20 0.43
HDAC1 Q13547 1/20 0.43
HDAC7 Q8WUI4 1/20 0.43
HDAC2 Q92769 1/20 0.43
HDAC10 Q969S8 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17927663 0.84 HTR6 (0.52) HTR6KDM4EUBE2NLMNASMN1; SMN2
SCHEMBL17927585 0.84 HTR6 (0.54) HTR6KDM4EUBE2NCA12CA9
SCHEMBL29651100 0.82 HTR6 (0.64) HTR6AKR1C3AKR1C1CA12CA9
SCHEMBL1996382 0.82 HTR6 (0.64) HTR6AKR1C3AKR1C1CA12CA9
SCHEMBL1015250 0.81 HTR6 (0.58) HTR6AKR1C3AKR1C1CA12CA9
SCHEMBL4334765 0.81 HTR6 (0.52) HTR6AKR1C3AKR1C1CA12CA9
SCHEMBL19737423 0.81 HTR6 (0.59) HTR6AKR1C3AKR1C1CA12CA9
SCHEMBL4334870 0.77 HTR6 (0.65) HTR6MEN1KMT2AHTR1ADRD2
SCHEMBL1156134 0.77 PARL (0.42) HTR6KDM4EUBE2NAKR1C3AKR1C1
SCHEMBL4781429 0.76 HTR6 (0.51) HTR6KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017216732-A1 AZA-TANSHINONE DERIVATIVES, PROCESS FOR THEIR PREPARATION AND THEIR USE IN THERAPY UNIVERSITA' DEGLI STUDI DI MILANO (IT) 2017-12-21 WO disclosed