SCHEMBL19742665

SCHEMBL19742665

CN(Cc1ccccc1)C(=O)C(C)(C)NC(=O)O

nearest known ligand 0.64

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 2/20 0.64
RAB9A P51151 4/20 0.59
NPC1 O15118 3/20 0.59
CA12 O43570 1/20 0.54
CA9 Q16790 1/20 0.54
KMT2A Q03164 4/20 0.51
MTOR P42345 1/20 0.50
MEN1 O00255 2/20 0.49
HPGD P15428 2/20 0.47
ABCC1 P33527 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30279911 0.83 RIPK1 (0.64) RIPK1RAB9ANPC1CA12CA9
SCHEMBL19742566 0.83 CTSL (0.57) RIPK1RAB9ANPC1CA12CA9
SCHEMBL12265785 0.82 RIPK1 (0.72) RIPK1RAB9ANPC1CA12CA9
SCHEMBL30279914 0.79 RIPK1 (0.68) RIPK1RAB9ANPC1CA12CA9
SCHEMBL17882380 0.78 RIPK1 (1.00) RIPK1RAB9ANPC1CA12CA9
Hydrochloric Acid SCHEMBL6527015 0.78 RIPK1 (0.66) RIPK1RAB9ANPC1CA12CA9
SCHEMBL2316926 0.77 RIPK1 (0.65) RIPK1RAB9ANPC1CA12CA9
SCHEMBL4471691 0.77 NPC1 (0.50) RIPK1RAB9ANPC1CA12CA9
SCHEMBL28126713 0.76 RIPK1 (0.63) RIPK1RAB9ANPC1CA12CA9
SCHEMBL180384 0.76 NPC1 (0.73) RIPK1RAB9ANPC1CA12CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3474855-B1 CK2 INHIBITORS, COMPOSITIONS AND METHODS THEREOF POLARIS PHARMACEUTICALS INC (US) 2022-01-26 EP disclosed
EP-3474855-A1 CK2 INHIBITORS, COMPOSITIONS AND METHODS THEREOF Polaris Pharmaceuticals, Inc. (US) 2019-05-01 EP disclosed
US-10227344-B2 CK2 inhibitors, compositions and methods thereof POLARIS PHARMACEUTICALS, INC. (US) 2019-03-12 US disclosed
WO-2017223432-A1 CK2 INHIBITORS, COMPOSITIONS AND METHODS THEREOF POLARIS PHARMACEUTICALS (US) 2017-12-28 WO disclosed
US-20170369489-A1 CK2 INHIBITORS, COMPOSITIONS AND METHODS THEREOF POLARIS PHARMACEUTICALS 2017-12-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170369489-A1 CK2 INHIBITORS, COMPOSITIONS AND METHODS THEREOF CSNK1A1, CSNK2A1, CSNK2A3 RIPK1 2132/4885RAB9A 3927/4885NPC1 4261/4885
US-10227344-B2 CK2 inhibitors, compositions and methods thereof CSNK1A1, CSNK2A1, CSNK2A3 RIPK1 2132/4885RAB9A 3927/4885NPC1 4261/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.