SCHEMBL19746414

SCHEMBL19746414

Cc1ccn(CCc2ccccc2)c(=O)n1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
CASR P41180 3/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.42
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HSD17B10 Q99714 1/20 0.42
MAPT P10636 1/20 0.42
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
MGLL Q99685 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
TDP2 O95551 1/20 0.41
HTT P42858 1/20 0.41
POLB P06746 1/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17554285 0.81 EP300 (0.44) P2RX7KMT2AMEN1ALDH1A1GSK3A
SCHEMBL19746431 0.77 GRM2 (0.41) P2RX7KMT2AMEN1ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL6011092 0.75 HSD17B10 (0.51) KMT2AALDH1A1KDM4ELMNATSHR
SCHEMBL19747231 0.74 HTT (0.39) P2RX7KMT2AALDH1A1KDM4ELMNA
SCHEMBL19747232 0.74 HTT (0.39) P2RX7KMT2AALDH1A1KDM4ELMNA
SCHEMBL2865257 0.73 KMT2A (0.40) KMT2AMEN1ALDH1A1KDM4ELMNA
SCHEMBL19746869 0.73 L3MBTL1 (0.39) P2RX7KMT2ACASRKDM4EGSK3A
SCHEMBL19746867 0.73 NOS1 (0.39) P2RX7KMT2AMEN1ALDH1A1KDM4E
SCHEMBL19746868 0.73 NOS1 (0.39) P2RX7KMT2AMEN1ALDH1A1KDM4E
SCHEMBL591865 0.72 DRD2 (0.44) KMT2AALDH1A1KDM4ELMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017222952-A1 3- HETEROARYL SUBSTITUTED 5-TRIFLUOROMETHYL OXADIAZOLES AS HISTONE DEACETYLASE 6 (HDAC6) INHIBITORS MERCK SHARP & DOHME CORP. (US) 2017-12-28 WO disclosed