SCHEMBL19746474

SCHEMBL19746474

N#Cc1cnn(Cc2ccccc2)c(=O)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.49
TSHR P16473 3/20 0.45
RECQL P46063 1/20 0.44
HTR2C P28335 2/20 0.44
HTR2B P41595 1/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
PKM P14618 2/20 0.44
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
HSD17B10 Q99714 2/20 0.43
MAPT P10636 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ADORA2A P29274 1/20 0.40
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
PKLR P30613 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8784355 0.78 PTGS1 (0.53) PTGS1TSHRRECQLHTR2CHTR2B
SCHEMBL19286604 0.76 TSHR (0.53) PTGS1TSHRRECQLALDH1A1LMNA
SCHEMBL1691731 0.76 PTGS1 (0.52) PTGS1TSHRRECQLHTR2CHTR2B
SCHEMBL8783376 0.76 PTGS1 (0.56) PTGS1TSHRRECQLHTR2CHTR2B
SCHEMBL17582636 0.75 PTGS1 (0.54) PTGS1TSHRRECQLHTR2CHTR2B
SCHEMBL20443987 0.73 PTGS1 (0.49) PTGS1TSHRRECQLHTR2CHTR2B
SCHEMBL17595809 0.73 PTGS1 (0.52) PTGS1TSHRRECQLHTR2CHTR2B
SCHEMBL18790701 0.72 RECQL (0.48) PTGS1TSHRRECQLALDH1A1HTT
SCHEMBL17582620 0.72 PTGS1 (0.57) PTGS1TSHRRECQLALDH1A1LMNA
SCHEMBL6233458 0.72 MAPK14 (0.57) PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017222952-A1 3- HETEROARYL SUBSTITUTED 5-TRIFLUOROMETHYL OXADIAZOLES AS HISTONE DEACETYLASE 6 (HDAC6) INHIBITORS MERCK SHARP & DOHME CORP. (US) 2017-12-28 WO disclosed