SCHEMBL19746594

SCHEMBL19746594

C[C@H](O)CCN(C)Cc1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 1/20 0.56
PRMT6 Q96LA8 1/20 0.56
PRMT8 Q9NR22 1/20 0.56
SIGMAR1 Q99720 1/20 0.51
TSHR P16473 3/20 0.47
ALDH1A1 P00352 2/20 0.47
SMN1; SMN2 Q16637 2/20 0.46
MAOB P27338 2/20 0.46
LMNA P02545 2/20 0.46
ADRA2B P18089 1/20 0.46
ADRA2C P18825 1/20 0.46
SLC6A2 P23975 1/20 0.46
HTR2A P28223 1/20 0.46
SLC6A4 P31645 1/20 0.46
ADRA1A P35348 1/20 0.46
OPRK1 P41145 1/20 0.46
SLC6A3 Q01959 1/20 0.46
KCNH2 Q12809 1/20 0.46
USP2 O75604 1/20 0.46
CYP3A4 P08684 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5478551 1.00 CARM1 (0.56) CARM1PRMT6PRMT8SIGMAR1TSHR
SCHEMBL8399769 0.89 SIGMAR1 (0.57) CARM1PRMT6PRMT8SIGMAR1MAOB
SCHEMBL4798287 0.86 CARM1 (0.53) CARM1PRMT6PRMT8SIGMAR1TSHR
SCHEMBL14578374 0.85 CARM1 (0.60) CARM1PRMT6PRMT8SIGMAR1TSHR
SCHEMBL27376496 0.84 TSHR (0.51) CARM1PRMT6PRMT8TSHRALDH1A1
SCHEMBL16653971 0.83 OPRK1 (0.45) CARM1PRMT6PRMT8TSHRALDH1A1
SCHEMBL5482899 0.83 CARM1 (0.50) CARM1PRMT6PRMT8SIGMAR1TSHR
SCHEMBL9788223 0.83 CARM1 (0.59) CARM1PRMT6PRMT8SIGMAR1TSHR
SCHEMBL4802584 0.83 CARM1 (0.50) CARM1PRMT6PRMT8SIGMAR1TSHR
SCHEMBL4852041 0.82 CARM1 (0.53) CARM1PRMT6PRMT8SIGMAR1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3472148-A1 CARBAMOYLOXYMETHYL TRIAZOLE CYCLOHEXYL ACIDS AS LPA ANTAGONISTS Bristol-Myers Squibb Company (US) 2019-04-24 EP disclosed
WO-2017223016-A1 CARBAMOYLOXYMETHYL TRIAZOLE CYCLOHEXYL ACIDS AS LPA ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 2017-12-28 WO disclosed